SCHEMBL14747016

SCHEMBL14747016

Nc1cc(Cl)c(-c2c(F)cccc2F)c(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.44
CYP3A4 P08684 5/20 0.42
ALDH1A1 P00352 3/20 0.42
TAAR1 Q96RJ0 1/20 0.39
TSHR P16473 1/20 0.39
TP53 P04637 1/20 0.39
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CASP1 P29466 1/20 0.35
RECQL P46063 1/20 0.35
GAA P10253 3/20 0.33
HTT P42858 2/20 0.33
SMARCA2 P51531 2/20 0.33
SMARCA4 P51532 2/20 0.33
PBRM1 Q86U86 2/20 0.33
ALOX15 P16050 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
LMNA P02545 1/20 0.33
MAPK1 P28482 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16013714 0.79 CYP3A4 (0.39) THRBCYP3A4ALDH1A1TSHRTP53
SCHEMBL1353155 0.78 THRB (0.67) THRBCYP3A4ALDH1A1TSHRTP53
SCHEMBL14744204 0.74 MAP2 (0.39) THRBCYP3A4ALDH1A1TAAR1TSHR
SCHEMBL12480139 0.72 MAOA (0.45) CYP3A4ALDH1A1TAAR1CA1CA2
SCHEMBL14744163 0.70 CYP3A4 (0.42) THRBCYP3A4ALDH1A1TAAR1TSHR
SCHEMBL3395334 0.69 NPC1 (0.37) TAAR1CA1CA2GAASMARCA2
SCHEMBL14746573 0.68 CYP3A4 (0.46) THRBCYP3A4ALDH1A1TAAR1TSHR
SCHEMBL4844609 0.68 THRB (0.68) THRBCYP3A4ALDH1A1TSHRTP53
SCHEMBL1029756 0.68 CYP3A4 (0.58) THRBCYP3A4ALDH1A1TSHRTP53
SCHEMBL4653575 0.67 PLA2G7 (0.42) CYP3A4ALDH1A1TAAR1TSHRTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013029338-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2013-03-07 WO disclosed