SCHEMBL14744340

SCHEMBL14744340

N#Cc1cc(N)cc(Cl)c1Br

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.41
ALDH1A1 P00352 3/20 0.41
THRB P10828 1/20 0.38
KDM4E B2RXH2 4/20 0.38
MAPT P10636 3/20 0.38
HPGD P15428 2/20 0.38
MEN1 O00255 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 1/20 0.38
USP2 O75604 1/20 0.36
TRPV4 Q9HBA0 1/20 0.35
KHK P50053 1/20 0.35
LMNA P02545 1/20 0.34
CSNK1A1 P48729 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
TSHR P16473 1/20 0.33
TP53 P04637 1/20 0.32
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2435542 0.78 CYP3A4 (0.56) CYP3A4ALDH1A1THRBKDM4EMAPT
SCHEMBL29054114 0.78 GPR35 (0.41) CYP3A4ALDH1A1KDM4EMAPTHPGD
SCHEMBL4515950 0.77 CYP3A4 (0.42) CYP3A4ALDH1A1THRBKDM4EMAPT
SCHEMBL1810042 0.77 ALDH1A1 (0.58) CYP3A4ALDH1A1THRBMAPTHPGD
SCHEMBL15274595 0.76 ALDH1A1 (0.38) CYP3A4ALDH1A1THRBKDM4EMAPT
SCHEMBL792557 0.75 TRPV4 (0.35) ALDH1A1TRPV4KHKVCAM1
SCHEMBL15277639 0.75 ALDH1A1 (0.41) CYP3A4ALDH1A1THRBKDM4EMAPT
SCHEMBL14744326 0.75 KHK (0.39) CYP3A4ALDH1A1KDM4EMAPTHPGD
SCHEMBL21051816 0.75 KDM4E (0.40) CYP3A4ALDH1A1KDM4EMAPTHPGD
SCHEMBL16236615 0.75 KHK (0.43) CYP3A4ALDH1A1THRBKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013029338-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2013-03-07 WO disclosed