SCHEMBL14745931

SCHEMBL14745931

O=C(O)Nc1nc(Cl)c2cccn2n1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 3/20 0.37
EPHB3 P54753 4/20 0.35
ADORA3 P0DMS8 3/20 0.35
ADORA2A P29274 3/20 0.35
RIPK2 O43353 1/20 0.35
LCK P06239 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HTT P42858 1/20 0.34
SPR P35270 2/20 0.34
JAK3 P52333 3/20 0.33
BTK Q06187 3/20 0.33
ADORA1 P30542 2/20 0.33
LMNA P02545 1/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
TTK P33981 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14757972 0.84 TGFBR1 (0.39) TDP2KDM4EALDH1A1JAK3BTK
SCHEMBL12066293 0.75 TGFBR1 (0.42) ADORA3KDM4EALDH1A1HTTJAK3
SCHEMBL14745860 0.74 MAPT (0.38) ADORA2AALDH1A1ADORA1LMNAJAK2
SCHEMBL19226350 0.74 JAK2 (0.53) KDM4EALDH1A1JAK3LMNAJAK2
SCHEMBL12395227 0.72 NUDT1 (0.47) ADORA2AJAK3ADORA1JAK2JAK1
SCHEMBL20839881 0.70 TDP2 (0.56) TDP2EPHB3HTTJAK3LMNA
SCHEMBL12395226 0.68 TGFBR1 (0.34) ADORA3ADORA2AADORA1
SCHEMBL21439130 0.67 SPR (0.44) EPHB3ADORA2AALDH1A1SPRADORA1
SCHEMBL13676572 0.66 AURKA (0.39) JAK3JAK2TTK
SCHEMBL12345323 0.66 AURKA (0.39) JAK3JAK2TTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013033093-A1 HETEROCYCLIC COMPOUNDS AS JANUS KINASE INHIBITORS BIOCRYST PHARMACEUTICALS, INC. (US) 2013-03-07 WO disclosed