SCHEMBL14747018

SCHEMBL14747018

O=[N+]([O-])c1cc(OC(F)(F)F)c(-c2ccccc2)c(-n2cccc2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
TDP1 Q9NUW8 5/20 0.38
PSD A5PKW4 2/20 0.35
KCNQ3 O43525 1/20 0.35
KCNQ2 O43526 1/20 0.35
LMNA P02545 1/20 0.34
F2RL3 Q96RI0 1/20 0.34
MAPT P10636 3/20 0.34
HTT P42858 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
SERPINE1 P05121 1/20 0.33
JAK2 O60674 1/20 0.33
TYK2 P29597 1/20 0.33
RECQL P46063 1/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14746790 0.78 ALDH1A1 (0.38) LMNAGAA
SCHEMBL29074273 0.72 RAB9A (0.54) AKR1C3AKR1C2MEN1KMT2A
SCHEMBL28456552 0.72 RORC (0.43) LMNA
SCHEMBL8531927 0.72 CYP19A1 (0.43) TDP1LMNAMAPTMEN1KMT2A
SCHEMBL28529302 0.67 EPAS1 (0.37) AKR1C3AKR1C2TDP1LMNAMAPT
SCHEMBL9367150 0.66 AKR1C3 (0.50) AKR1C3AKR1C2TDP1LMNAMAPT
SCHEMBL14746841 0.66 PTGS2 (0.50) AKR1C3AKR1C2MAPTMEN1KMT2A
SCHEMBL1360458 0.64 PSD (0.39) AKR1C3AKR1C2PSDMAPTMEN1
SCHEMBL16923592 0.64 HTT (0.62) AKR1C3AKR1C2TDP1MAPTHTT
SCHEMBL1744862 0.64 ALDH1A1 (0.53) TDP1LMNAMAPTHTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013029338-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2013-03-07 WO disclosed