SCHEMBL1476924

SCHEMBL1476924

CON(C)C(=O)C1(C)CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HPGD P15428 1/20 0.38
EPHX2 P34913 1/20 0.38
RECQL P46063 1/20 0.37
EPHX1 P07099 1/20 0.37
ALDH1A1 P00352 2/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
NR1H2 P55055 1/20 0.36
GPR119 Q8TDV5 1/20 0.36
TSHR P16473 2/20 0.36
ALOX15 P16050 1/20 0.36
ATM Q13315 1/20 0.36
USP30 Q70CQ3 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22164606 0.92 USP2 (0.39) USP2SMN1; SMN2HPGDEPHX2NR1H2
SCHEMBL17848733 0.86 USP2 (0.47) USP2SMN1; SMN2HPGDEPHX2RECQL
SCHEMBL23249895 0.85 USP2 (0.44) USP2SMN1; SMN2HPGDEPHX2RECQL
SCHEMBL25309715 0.85 USP2 (0.39) USP2SMN1; SMN2HPGDEPHX2RECQL
SCHEMBL1475506 0.84 USP30 (0.43) USP2SMN1; SMN2HPGDEPHX2RECQL
SCHEMBL26316172 0.83 HPGD (0.38) USP2SMN1; SMN2HPGDEPHX2EPHX1
SCHEMBL16987667 0.82 USP2 (0.41) USP2SMN1; SMN2HPGDEPHX2GPR119
SCHEMBL21807050 0.81 USP2 (0.40) USP2SMN1; SMN2HPGDEPHX2RECQL
SCHEMBL29959181 0.79 USP30 (0.51) USP2SMN1; SMN2HPGDNR1H2USP30
SCHEMBL23578737 0.79 USP30 (0.51) USP2SMN1; SMN2HPGDNR1H2USP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233077-B1 DOPAMINE D2 RECEPTOR LIGANDS BROAD INST INC (US) 2026-05-06 EP disclosed
EP-4720041-A2 N-(1H-INDOL-2-YL)METHYL)-4-ETHYNYL-PICOLINAMIDE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER Allorion Therapeutics Inc (US) 2026-04-08 EP disclosed
US-12428373-B2 Dopamine D2 receptor ligands THE BROAD INSTITUTE, INC. (US) 2025-09-30 US disclosed
US-20250026763-A1 EGFR INHIBITORS AND METHODS OF USE THEREOF Allorion Therapeutics Inc 2025-01-23 US disclosed
WO-2024240241-A2 EGFR INHIBITORS AND METHODS OF USE THEREOF Allorion Therapeutics Inc (US) 2024-11-28 WO disclosed
US-11932643-B2 Substituted heterocyclic inhibitors of PTPN11 NAVIRE PHARMA, INC. (US) 2024-03-19 US disclosed
US-11840536-B2 Heterocyclic inhibitors of PTPN11 BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2023-12-12 US disclosed
CN-112351780-B Substituted heterocyclic inhibitors of PTPN11 纳维尔制药有限公司 2023-12-01 CN disclosed
CN-114127053-B Substituted pyrazine compound, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2023-06-13 CN disclosed
US-20230143552-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2023-05-11 US disclosed
EP-3233077-A1 DOPAMINE D2 RECEPTOR LIGANDS The Broad Institute Inc. (US) 2017-10-25 EP disclosed
WO-2016100940-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2016-06-23 WO disclosed
US-20130345215-A1 PYRAZOLOPYRIMIDONE AND PYRAZOLOPYRIDONE INHIBITORS OF TANKYRASE F. HOFFMANN-LA ROCHE AG (CH) 2013-12-26 US disclosed
US-7915274-B2 Nitrogen containing heterocyclic compounds and medicines containing the same EISAI R&D MANAGEMENT CO., LTD. (JP) 2011-03-29 US disclosed
US-20070293496-A1 Nitrogen containing heterocyclic compounds and medicines containing the same OZAKI FUMIHIRO 2007-12-20 US disclosed
US-7265108-B2 Nitrogen containing heterocyclic compounds and medicines containing the same EISAI CO., LTD. (JP) 2007-09-04 US disclosed
EP-1484327-B1 NITROGENOUS HETEROCYCLIC COMPOUND AND MEDICINE THEREOF EISAI R&D MAN CO LTD (JP) 2007-08-01 EP disclosed
US-6995144-B2 Nitrogen containing heterocyclic compounds and medicines containing the same EISAI CO., LTD. (JP) 2006-02-07 US disclosed
US-20050245527-A1 Nitrogen containing heterocyclic compounds and medicines containing the same EISAI R&D MANAGEMENT CO., LTD. (JP) 2005-11-03 US disclosed
EP-1484327-A1 NITROGENOUS HETEROCYCLIC COMPOUND AND MEDICINE THEREOF Eisai Co., Ltd. (JP) 2004-12-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070293496-A1 Nitrogen containing heterocyclic compounds and medicines containing the same XDH, NQO1, CYP1A1 USP2 3639/4885SMN1; SMN2 1451/4885HPGD 147/4885
US-20230143552-A1 DOPAMINE D2 RECEPTOR LIGANDS DRD2, SLC6A3, NTSR2 USP2 1115/4885SMN1; SMN2 1443/4885HPGD 2049/4885
US-12428373-B2 Dopamine D2 receptor ligands DRD2, SLC6A3, NTSR2 USP2 1115/4885SMN1; SMN2 1443/4885HPGD 2049/4885
US-11932643-B2 Substituted heterocyclic inhibitors of PTPN11 PTPN11, PTPRJ, PTPRCAP USP2 1009/4885SMN1; SMN2 4080/4885HPGD 1873/4885
US-20130345215-A1 PYRAZOLOPYRIMIDONE AND PYRAZOLOPYRIDONE INHIBITORS OF TANKYRASE TNKS1BP1, TPI1, TNKS USP2 2161/4885SMN1; SMN2 3043/4885HPGD 1462/4885
US-20250026763-A1 EGFR INHIBITORS AND METHODS OF USE THEREOF EGFR, ERBB3, ERBB2 USP2 1727/4885SMN1; SMN2 4856/4885HPGD 4268/4885
US-11840536-B2 Heterocyclic inhibitors of PTPN11 PTPRJ, PTPN11, PTPRCAP USP2 1045/4885SMN1; SMN2 4183/4885HPGD 1782/4885
US-20050245527-A1 Nitrogen containing heterocyclic compounds and medicines containing the same XDH, NQO1, CYP1A1 USP2 3639/4885SMN1; SMN2 1451/4885HPGD 147/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.