Lonazolac

Lonazolac

SCHEMBL1478078

O=C(O)Cc1cn(-c2ccccc2)nc1-c1ccc(Cl)cc1.O=C(O)Cc1cn(-c2ccccc2)nc1-c1ccc(Cl)cc1.[CaH2]

nearest known ligand 0.97

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.97
DRD2 P14416 1/20 0.97
PTGES O14684 9/20 0.84
ALOX5 P09917 8/20 0.84
ALDH1A1 P00352 3/20 0.80
AGTR1 P30556 1/20 0.64
KMT2A Q03164 1/20 0.64
CCNE1 P24864 3/20 0.62
CDK2 P24941 3/20 0.62
MAPT P10636 2/20 0.59
HPGD P15428 2/20 0.59
USP2 O75604 1/20 0.59
NPSR1 Q6W5P4 1/20 0.59
HSD17B10 Q99714 1/20 0.59
AURKA O14965 2/20 0.57
LMNA P02545 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lonazolac SCHEMBL287156 1.00 KDM4E (0.97) KDM4EDRD2PTGESALOX5ALDH1A1
Lonazolac SCHEMBL25221 0.99 KDM4E (1.00) KDM4EDRD2PTGESALOX5ALDH1A1
SCHEMBL11245260 0.93 KDM4E (0.90) KDM4EDRD2PTGESALOX5ALDH1A1
SCHEMBL11166545 0.93 KDM4E (0.90) KDM4EDRD2PTGESALOX5ALDH1A1
SCHEMBL10877279 0.90 KDM4E (0.83) KDM4EDRD2PTGESALOX5ALDH1A1
SCHEMBL10407060 0.89 KDM4E (1.00) KDM4EDRD2PTGESALOX5ALDH1A1
SCHEMBL12608902 0.88 KDM4E (0.81) KDM4EDRD2PTGESALOX5ALDH1A1
SCHEMBL3475488 0.88 KDM4E (0.81) KDM4EDRD2PTGESALOX5ALDH1A1
Lonazolac SCHEMBL10577835 0.87 PTGES (1.00) KDM4EDRD2PTGESALOX5ALDH1A1
SCHEMBL11258042 0.87 KDM4E (0.79) KDM4EDRD2PTGESALOX5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752201-B1 SUSPENSION OF NANOSCALE, ORGANIC PARTICLES AND PROCESS FOR PRODUCTION THEREOF UNIV FRIEDRICH ALEXANDER ER (DE) 2023-11-22 EP disclosed
EP-3752201-A1 SUSPENSION OF NANOSCALE, ORGANIC PARTICLES AND PROCESS FOR PRODUCTION THEREOF Friedrich-Alexander-Universität Erlangen-Nürnberg (DE) 2020-12-23 EP disclosed
US-9023889-B2 Use of ascorbic acid derivatives for the functionalization of matrices MERCK PATENT GMBH (DE) 2015-05-05 US disclosed
EP-1860158-B1 Particles comprising a substrate and an anion-binding layer MERCK PATENT GMBH (DE) 2013-12-04 EP disclosed
US-7927613-B2 Pharmaceutical co-crystal compositions UNIVERSITY OF SOUTH FLORIDA (US) 2011-04-19 US disclosed
US-7914893-B2 Particles comprising an anion-binding layer containing anion-forming organic active compounds, and method of making and using thereof MERCK PATENT GMBH (DE) 2011-03-29 US disclosed
US-7790905-B2 Pharmaceutical propylene glycol solvate compositions MCNEIL-PPC, INC. (US) 2010-09-07 US disclosed
US-20100167936-A1 USE OF ASCORBIC ACID DERIVATIVES FOR THE FUNCTIONALIZATION OF MATRICES MERCK PATENT GESELLSCHAFT (DE) 2010-07-01 US disclosed
EP-2049075-A2 USE OF ASCORBIC ACID DERIVATIVES FOR THE FUNCTIONALIZATION OF MATRICES Merck Patent GmbH (DE) 2009-04-22 EP disclosed
WO-2008017346-A2 USE OF ASCORBIC ACID DERIVATIVES FOR THE FUNCTIONALIZATION OF MATRICES MERCK PATENT GMBH (DE) 2008-02-14 WO disclosed
US-20070275244-A1 Particles MERCK PATENT GMBH 2007-11-29 US disclosed
EP-1860158-A2 Particles comprising a substrate and an anion-binding layer MERCK PATENT GmbH (DE) 2007-11-28 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100167936-A1 USE OF ASCORBIC ACID DERIVATIVES FOR THE FUNCTIONALIZATION OF MATRICES PROC, TTPA, COX6C KDM4E 4007/4885DRD2 1441/4885PTGES 2360/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.