SCHEMBL14782827

SCHEMBL14782827

COC(=O)c1cc(CNC(=O)C2CCC2)ccc1Cl

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 1/20 0.53
ERCC4 Q92889 1/20 0.53
HPGD P15428 6/20 0.53
LMNA P02545 2/20 0.53
ALDH1A1 P00352 4/20 0.51
USP2 O75604 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.49
TSHR P16473 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
EPHX2 P34913 1/20 0.47
NPC1 O15118 1/20 0.46
PKM P14618 1/20 0.46
RAB9A P51151 1/20 0.46
HDAC6 Q9UBN7 1/20 0.45
KDM4E B2RXH2 2/20 0.44
ALOX15 P16050 1/20 0.44
KCNH2 Q12809 1/20 0.43
HTR4 Q13639 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14782977 0.95 HPGD (0.55) ERCC1ERCC4HPGDLMNAALDH1A1
Hydrochloric Acid SCHEMBL25251752 0.88 HPGD (0.49) ERCC1ERCC4HPGDLMNAALDH1A1
SCHEMBL14783181 0.86 ALDH1A1 (0.58) ERCC1ERCC4HPGDLMNAALDH1A1
SCHEMBL14782820 0.85 LMNA (0.48) ERCC1ERCC4HPGDLMNAALDH1A1
SCHEMBL14782775 0.82 PKM (0.55) HPGDLMNAALDH1A1SMN1; SMN2TSHR
SCHEMBL30491752 0.80 ERCC1 (0.52) ERCC1ERCC4HPGDLMNAALDH1A1
SCHEMBL14782772 0.80 ERCC1 (0.52) ERCC1ERCC4HPGDLMNAALDH1A1
SCHEMBL18810198 0.77 ERCC1 (0.49) ERCC1ERCC4HPGDLMNAALDH1A1
SCHEMBL16992006 0.77 NPC1 (0.62) ERCC1ERCC4HPGDLMNAALDH1A1
SCHEMBL14783152 0.77 LMNA (0.55) HPGDLMNAALDH1A1SMN1; SMN2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013038308-A1 SUBSTITUTED BICYCLIC HETEROARYL COMPOUNDS AS mPGES-1 INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2013-03-21 WO disclosed
WO-2013038308-A1 SUBSTITUTED BICYCLIC HETEROARYL COMPOUNDS AS mPGES-1 INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2013-03-21 WO disclosed