SCHEMBL1478638

SCHEMBL1478638

CN(Cc1ccc(C(=O)O[Si](C)(C)C)cc1)[Si](C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 1/20 0.38
ALDH1A1 P00352 5/20 0.37
SMN1; SMN2 Q16637 4/20 0.37
HPGD P15428 3/20 0.37
KDM4E B2RXH2 2/20 0.37
NPC1 O15118 2/20 0.37
GAA P10253 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
HSD17B10 Q99714 1/20 0.37
RAB9A P51151 2/20 0.36
MAPT P10636 3/20 0.36
PYCR1 P32322 1/20 0.36
POLB P06746 1/20 0.36
ACHE P22303 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
CYP4A11 Q02928 1/20 0.35
HSP90AA1 P07900 1/20 0.34
HDAC8 Q9BY41 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1478927 0.87 LOXL2 (0.40) LOXL2ALDH1A1SMN1; SMN2HPGDKDM4E
SCHEMBL1479438 0.81 ALDH1A1 (0.31) ALDH1A1SMN1; SMN2MAPTPYCR1POLB
SCHEMBL11897476 0.80 ALDH1A1 (0.52) ALDH1A1SMN1; SMN2HPGDKDM4EGAA
SCHEMBL8460883 0.78 CA1 (0.44) LOXL2ALDH1A1HPGDKDM4EGAA
SCHEMBL1478516 0.78 ALDH1A1 (0.38) ALDH1A1SMN1; SMN2HPGDKDM4ENPC1
SCHEMBL12212913 0.73 PDCD1 (0.46) ALDH1A1SMN1; SMN2HPGDKDM4ENPC1
SCHEMBL11897625 0.73 ALDH1A1 (0.37) ALDH1A1SMN1; SMN2HPGDTSHRMAPT
SCHEMBL1478754 0.73 NOTUM (0.36) ALDH1A1SMN1; SMN2HPGDKDM4ENPC1
SCHEMBL10917868 0.71 HPGD (0.54) ALDH1A1SMN1; SMN2HPGDTSHRMAPT
SCHEMBL10931509 0.71 CA12 (0.59) ALDH1A1SMN1; SMN2HPGDNPC1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895670-B2 Functionalized polymers and methods for their manufacture BRIDGESTONE CORPORATION (JP) 2014-11-25 US claimed
US-20110077325-A1 FUNCTIONALIZED POLYMERS AND METHODS FOR THEIR MANUFACTURE BRIDGESTONE CORPORATION (JP) 2011-03-31 US claimed
EP-2699606-B1 POLYMERS FUNCTIONALIZED WITH A CARBOXYLIC OR THIOCARBOXYLIC ESTER CONTAINING A SILYLATED AMINO GROUP BRIDGESTONE CORP (JP) 2016-09-28 EP disclosed
US-9403919-B2 Polymers functionalized with a carboxylic or thiocarboxylic ester containing a silylated amino group BRIDGESTONE CORPORATION (JP) 2016-08-02 US disclosed
US-8895670-B2 Functionalized polymers and methods for their manufacture BRIDGESTONE CORPORATION (JP) 2014-11-25 US disclosed
EP-2699606-A2 POLYMERS FUNCTIONALIZED WITH A CARBOXYLIC OR THIOCARBOXYLIC ESTER CONTAINING A SILYLATED AMINO GROUP Bridgestone Corporation (JP) 2014-02-26 EP disclosed
EP-2483317-B1 FUNCTIONALIZED POLYMERS AND METHODS FOR THEIR MANUFACTURE BRIDGESTONE CORP (JP) 2014-02-26 EP disclosed
US-20140018500-A1 Polymers Functionalized With A Carboxylic Or Thiocarboxylic Ester Containing A Silylated Amino Group BRIDGESTONE CORPORATION (JP) 2014-01-16 US disclosed
WO-2012135451-A2 POLYMERS FUNCTIONALIZED WITH A CARBOXYLIC OR THIOCARBOXYLIC ESTER CONTAINING A SILYLATED AMINO GROUP BRIDGESTONE CORPORATION (JP) 2012-10-04 WO disclosed
US-20120184677-A1 FUNCTIONALIZED POLYMERS AND METHODS FOR THEIR MANUFACTURE BRIDGESTONE CORPORATION (JP) 2012-07-19 US disclosed
US-20110077325-A1 FUNCTIONALIZED POLYMERS AND METHODS FOR THEIR MANUFACTURE BRIDGESTONE CORPORATION (JP) 2011-03-31 US disclosed