SCHEMBL14795178

SCHEMBL14795178

CC(C)(C)OC(=O)ON1CCC(Oc2ccc(OCC(F)(F)F)cc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACACB O00763 8/20 0.49
LIPE Q05469 3/20 0.46
MMP13 P45452 1/20 0.46
MMP14 P50281 1/20 0.46
GPR119 Q8TDV5 3/20 0.44
SCN9A Q15858 1/20 0.42
CARM1 Q86X55 1/20 0.40
PRMT6 Q96LA8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL75960 0.84 GPR119 (0.62) ACACBLIPEGPR119
SCHEMBL3724395 0.83 GPR119 (0.46) ACACBGPR119
SCHEMBL373517 0.83 GPR119 (0.46) ACACBGPR119
SCHEMBL373589 0.81 MAPT (0.42) GPR119
SCHEMBL7308360 0.80 GPR119 (0.44) ACACBGPR119
SCHEMBL14795180 0.80 ACACB (0.49) ACACBLIPEMMP13MMP14SCN9A
SCHEMBL14795181 0.76 HRH1 (0.43) ACACBLIPEMMP13MMP14GPR119
SCHEMBL74340 0.75 GPR119 (0.60) LIPEMMP13MMP14GPR119
SCHEMBL373986 0.74 ESR2 (0.49) GPR119
SCHEMBL7301874 0.74 POLB (0.42) ACACBGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2573090-B1 (6,7-DIHYDRO-2-NITRO-5H-IMIDAZOL[2,1-B][1,3]OXAZIN-6-YL) AMIDE COMPOUNDS, PREPARATION METHODS AND USES THEREOF SHANGHAI SUN SAIL PHARMACEUTICAL SCIENCE & TECHNOLOGY CO LTD (CN) 2014-12-10 EP disclosed
US-8563547-B2 (6,7-dihydro-2-nitro-5H-imidazol[2,1-b][1,3]oxazin-6-yl) amide compounds, preparation methods and uses thereof SHANGHAI SUN-SAIL PHARMACEUTICAL SCIENCE & TECHNOLOGY CO., LTD. (CN) 2013-10-22 US disclosed
US-20130143864-A1 (6,7-DIHYDRO-2-NITRO-5H-IMIDAZOL[2,1-B][1,3]OXAZIN-6YL) AMIDE COMPOUNDS, PREPARATION METHODS AND USES THEREOF NANJING CHANGAO PHARMACEUTICAL SCIENCE & TECHNOLOGY CO., LTD. (CN) 2013-06-06 US disclosed
EP-2573090-A1 (6,7-DIHYDRO-2-NITRO-5H-IMIDAZOL[2,1-B][1,3]OXAZIN-6-YL) AMIDE COMPOUNDS, PREPARATION METHODS AND USES THEREOF Shanghai Sun-Sail Pharmaceutical Science & Technology Co., Ltd (CN) 2013-03-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130143864-A1 (6,7-DIHYDRO-2-NITRO-5H-IMIDAZOL[2,1-B][1,3]OXAZIN-6YL) AMIDE COMPOUNDS, PREPARATION METHODS AND USES THEREOF MT-ND6, SLC11A2, NDUFB7 ACACB 754/4885LIPE 3617/4885MMP13 3963/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.