SCHEMBL14799727

SCHEMBL14799727

COC(=O)CCNC(=O)OC(C)(C)Cc1ccc(N)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
NFKB1 P19838 1/20 0.40
CYP2C19 P33261 1/20 0.40
LMNA P02545 1/20 0.39
PMP22 Q01453 1/20 0.39
NLRP3 Q96P20 1/20 0.39
ESRRG P62508 1/20 0.39
PPIB P23284 1/20 0.39
PPIA P62937 1/20 0.39
PPID Q08752 1/20 0.39
PPIG Q13427 1/20 0.39
CTSK P43235 3/20 0.39
EPHX2 P34913 1/20 0.38
CA2 P00918 3/20 0.38
CA1 P00915 2/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25342471 0.76 CYP3A4 (0.50) CYP3A4CYP1A2CYP2D6CYP2C9NFKB1
SCHEMBL16503439 0.75 CA12 (0.48) LMNAPPIBPPIAPPIDPPIG
SCHEMBL5000597 0.75 KMT2A (0.42) CYP3A4CYP1A2CYP2D6CYP2C9NFKB1
SCHEMBL5869428 0.74 HPGD (0.39) LMNAKDM4EALDH1A1GLAGAA
SCHEMBL15075046 0.74 POLB (0.56) LMNAKDM4EALDH1A1HPGD
SCHEMBL27495164 0.73 CYP3A4 (0.50) CYP3A4CYP1A2CYP2D6CYP2C9NFKB1
SCHEMBL448114 0.73 CA2 (0.58) LMNAESRRGCTSKCA2CA1
SCHEMBL1256643 0.72 TDP1 (0.55) EPHX2CA2CA1KDM4EALDH1A1
SCHEMBL2667533 0.72 LMNA (0.56) CYP1A2CYP2C19LMNAPMP22ESRRG
SCHEMBL3912645 0.72 CTSK (0.43) CTSKCA2CA1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130079383-A1 Lipid Compounds Targeting VLA-4 ARROWHEAD RESEARCH CORPORATION (US) 2013-03-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130079383-A1 Lipid Compounds Targeting VLA-4 LPAR4, ASGR1, VCAM1 CYP3A4 1386/4885CYP1A2 3014/4885CYP2D6 2343/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.