SCHEMBL14809682

SCHEMBL14809682

COc1cc(-c2nccn2C2CC2)cnc1F

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.39
CYP11B2 P19099 9/20 0.38
CYP11B1 P15538 7/20 0.38
GSK3B P49841 1/20 0.35
MAPK14 Q16539 1/20 0.34
GABRA2 P47869 2/20 0.33
KCNH2 Q12809 2/20 0.32
PIK3CA P42336 1/20 0.32
LRRK2 Q5S007 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20339238 0.73 CYP11B2 (0.50) CYP11B2CYP11B1
SCHEMBL28344812 0.69 CYP11B2 (0.55) CYP11B2CYP11B1
SCHEMBL28344944 0.69 CYP11B2 (0.56) CYP11B2CYP11B1
SCHEMBL27277040 0.67 PDE4A (0.44) MAPK14
SCHEMBL20339309 0.66 CYP11B1 (0.51) CYP11B2CYP11B1
SCHEMBL28226097 0.66 ESR1 (0.41) CYP11B2MAPK14
SCHEMBL4373862 0.64 ACHE (0.43)
SCHEMBL29698205 0.64 ACHE (0.43)
SCHEMBL15315959 0.64 LMNA (0.37)
SCHEMBL6039495 0.63 CYP1A2 (0.49) MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2757882-A1 IMIDAZOPYRIDYL COMPOUNDS AS ALDOSTERONE SYNTHASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2014-07-30 EP disclosed
WO-2013043518-A1 IMIDAZOPYRIDYL COMPOUNDS AS ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2013-03-28 WO disclosed