SCHEMBL14822757

SCHEMBL14822757

Fc1ccc(Cn2cccn2)c(F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.48
KDM4E B2RXH2 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
BRD4 O60885 1/20 0.46
KLKB1 P03952 1/20 0.43
HDAC1 Q13547 2/20 0.41
HDAC7 Q8WUI4 1/20 0.41
KAT7 O95251 1/20 0.40
KAT6B Q8WYB5 1/20 0.40
KAT6A Q92794 1/20 0.40
KAT5 Q92993 1/20 0.40
KAT8 Q9H7Z6 1/20 0.40
HTT P42858 1/20 0.40
IDO1 P14902 2/20 0.40
AGXT P21549 2/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
HTR2A P28223 1/20 0.38
BCHE P06276 1/20 0.37
ACHE P22303 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14822759 0.87 RIPK1 (0.44) CYP3A4BRD4HDAC1KAT7KAT6B
SCHEMBL3806937 0.84 SMN1; SMN2 (0.48) KDM4ESMN1; SMN2BRD4HTTGAA
SCHEMBL3809851 0.84 TP53 (0.45) CYP3A4BRD4KLKB1HDAC1HTT
SCHEMBL1953678 0.84 BRD4 (0.43) CYP3A4BRD4KLKB1HDAC1HTT
SCHEMBL5299707 0.84 BRD4 (0.43) CYP3A4KDM4ESMN1; SMN2BRD4KLKB1
SCHEMBL17221362 0.81 KLKB1 (0.47) CYP3A4BRD4KLKB1HDAC1KAT7
SCHEMBL30047375 0.81 ALDH1A1 (0.56) CYP3A4KDM4ESMN1; SMN2BRD4HDAC1
SCHEMBL7465706 0.81 ALDH1A1 (0.56) CYP3A4KDM4ESMN1; SMN2BRD4HDAC1
SCHEMBL27760047 0.80 KDM4E (0.49) KDM4ESMN1; SMN2BRD4KLKB1KAT7
SCHEMBL31691366 0.79 HTT (0.60) BRD4KLKB1HDAC1HDAC7HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103097387-B Ring-fused pyrimidines and triazines and use thereof for treating and/or preventing cardiovascular diseases 拜耳知识产权有限责任公司 2016-11-02 CN disclosed
EP-3048155-A1 ORGANIC MOLECULES, IN PARTICULAR FOR USE IN OPTOELECTRONIC COMPONENTS cynora GmbH (DE) 2016-07-27 EP disclosed
EP-3048156-A1 ORGANIC MOLECULES, IN PARTICULAR FOR USE IN OPTOELECTRONIC COMPONENTS cynora GmbH (DE) 2016-07-27 EP disclosed
CN-104011027-A Use of lonidamine analogs for fertility regulation UNIV KANSAS 2014-08-27 CN disclosed
CN-103097387-A Ring-fused pyrimidines and triazines and use thereof for treating and/or preventing cardiovascular diseases BAYER IP GMBH 2013-05-08 CN disclosed
US-8410269-B2 Phosphorescent iridium complex with non-conjugated cyclometalated ligands, synthetic method of preparing the same and phosphorescent organic light emitting diode thereof NATIONAL TSING HUA UNIVERSITY (TW) 2013-04-02 US disclosed
US-20110313162-A1 PHOSPHORESCENT IRIDIUM COMPLEX WITH NON-CONJUGATED CYCLOMETALATED LIGANDS, SYNTHETIC METHOD OF PREPARING THE SAME AND PHOSPHORESCENT ORGANIC LIGHT EMITTING DIODE THEREOF NATIONAL TSING HUA UNIVERSITY (TW) 2011-12-22 US disclosed
US-20110313161-A1 PHOSPHORESCENT IRIDIUM COMPLEX WITH NON-CONJUGATED CYCLOMETALATED LIGANDS, SYNTHETIC METHOD OF PREPARING THE SAME AND PHOSPHORESCENT ORGANIC LIGHT EMITTING DIODE THEREOF NATIONAL TSING HUA UNIVERSITY (TW) 2011-12-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110313161-A1 PHOSPHORESCENT IRIDIUM COMPLEX WITH NON-CONJUGATED CYCLOMETALATED LIGANDS, SYNTHETIC METHOD OF PREPARING THE SAME AND PHOSPHORESCENT ORGANIC LIGHT EMITTING DIODE THEREOF LIG3, LIG4, LIG1 CYP3A4 4333/4885KDM4E 3694/4885SMN1; SMN2 4318/4885
US-20110313162-A1 PHOSPHORESCENT IRIDIUM COMPLEX WITH NON-CONJUGATED CYCLOMETALATED LIGANDS, SYNTHETIC METHOD OF PREPARING THE SAME AND PHOSPHORESCENT ORGANIC LIGHT EMITTING DIODE THEREOF LIG3, LIG4, LIG1 CYP3A4 4333/4885KDM4E 3694/4885SMN1; SMN2 4318/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.