SCHEMBL1483632

SCHEMBL1483632

O=c1cc(-c2cc(OCc3ccccc3)cc(OCc3ccccc3)c2)oc2cc(O)ccc12

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.66
CYP19A1 P11511 2/20 0.66
MAOA P21397 2/20 0.66
MAOB P27338 2/20 0.66
AKR1B1 P15121 2/20 0.66
CALM1 P0DP23 2/20 0.66
PKM P14618 2/20 0.66
FTO Q9C0B1 2/20 0.66
CA12 O43570 1/20 0.66
AKR1B10 O60218 1/20 0.66
CA1 P00915 1/20 0.66
CA2 P00918 1/20 0.66
CYP1A2 P05177 1/20 0.66
HSD17B1 P14061 1/20 0.66
HSD17B3 P37058 1/20 0.66
XDH P47989 1/20 0.66
CYP1B1 Q16678 1/20 0.66
CA9 Q16790 1/20 0.66
MAPT P10636 2/20 0.62
CYP3A4 P08684 3/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4406405 0.84 SIGMAR1 (0.55) ABCB1MAOAMAOBMAPTL3MBTL1
SCHEMBL4157444 0.84 CYP19A1 (0.63) ABCB1CYP19A1MAOAMAOBAKR1B1
SCHEMBL28078087 0.84 MAOB (0.67) ABCB1CYP19A1MAOAMAOBAKR1B1
SCHEMBL12756579 0.82 ABCB1 (0.50) ABCB1MAOBMAPTL3MBTL1
SCHEMBL12756580 0.82 ABCB1 (0.50) ABCB1MAOBMAPTL3MBTL1
SCHEMBL1483628 0.82 PRKDC (0.52) ABCB1MAOAMAOBMAPTL3MBTL1
SCHEMBL1483630 0.82 PRKDC (0.52) ABCB1MAOAMAOBMAPTL3MBTL1
SCHEMBL1483626 0.82 PRKDC (0.52) ABCB1MAOAMAOBMAPTL3MBTL1
7-Hydroxyflavone SCHEMBL29678183 0.80 CYP19A1 (1.00) ABCB1CYP19A1MAOAMAOBAKR1B1
7-Hydroxyflavone SCHEMBL312148 0.80 CYP19A1 (1.00) ABCB1CYP19A1MAOAMAOBAKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1807408-B1 OXY SUBSTITUTED FLAVONES AS ANTIHYPERGLYCEMIC AND ANTIDYSLIPIDEMIC AGENTS COUNCIL SCIENT IND RES (IN) 2016-06-08 EP disclosed
EP-2057137-B1 S-(+)-7-[3-N-SUBSTITUTED AMINO-2-HYDROXYPROPOXY]FLAVONES COUNCIL SCIENT IND RES (IN) 2013-10-23 EP disclosed
US-20110077294-A1 R-(-) / S-(+)-7-[3-N SUBSTITUTED AMINO-2 HYDROXYPROPOXY] FLAVONES COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2011-03-31 US disclosed
US-20110077294-A1 R-(-) / S-(+)-7-[3-N SUBSTITUTED AMINO-2 HYDROXYPROPOXY] FLAVONES COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2011-03-31 US disclosed
US-7635779-B2 Oxy substituted flavones as antihyperglycemic and antidyslipidemic agents COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2009-12-22 US disclosed
EP-2057137-A1 R-(-) / S-(+)-7-[3-N-SUBSTITUTED AMINO-2-HYDROXYPROPOXY]FLAVONES Council of Scientific and Industrial Research (IN) 2009-05-13 EP disclosed
WO-2008018089-A1 R-(-) / S-(+)-7-[3-N-SUBSTITUTED AMINO-2-HYDROXYPROPOXY] FLAVONES COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2008-02-14 WO disclosed
WO-2008018089-A1 R-(-) / S-(+)-7-[3-N-SUBSTITUTED AMINO-2-HYDROXYPROPOXY] FLAVONES COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2008-02-14 WO disclosed
EP-1807408-A1 OXY SUBSTITUTED FLAVONES AS ANTIHYPERGLYCEMIC AND ANTIDYSLIPIDEMIC AGENTS Council of Scientific and Industrial Research (IN) 2007-07-18 EP disclosed
US-20060178373-A1 Oxy substituted flavones as antihyperglycemic and antidyslipidemic agents COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2006-08-10 US disclosed
WO-2006040621-A1 OXY SUBSTITUTED FLAVONES AS ANTIHYPERGLYCEMIC AND ANTIDYSLIPIDEMIC AGENTS COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2006-04-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110077294-A1 R-(-) / S-(+)-7-[3-N SUBSTITUTED AMINO-2 HYDROXYPROPOXY] FLAVONES HTR7, PNMT, PRMT7 ABCB1 944/4885CYP19A1 290/4885MAOA 333/4885
US-20060178373-A1 Oxy substituted flavones as antihyperglycemic and antidyslipidemic agents GPR119, LIPC, SLC5A2 ABCB1 1033/4885CYP19A1 151/4885MAOA 948/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.