SCHEMBL14844199

SCHEMBL14844199

Fc1cccc(F)c1C1CNc2cccnc2O1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
NISCH Q9Y2I1 1/20 0.34
LTA4H P09960 1/20 0.34
JAK2 O60674 1/20 0.34
AKT1 P31749 1/20 0.32
HTR1A P08908 2/20 0.32
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 1/20 0.32
P2RX7 Q99572 2/20 0.30
NOS3 P29474 1/20 0.30
NOS1 P29475 1/20 0.30
NOS2 P35228 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14844536 0.80 CHRNB2 (0.32) CHRNB2CHRNA4
SCHEMBL14845191 0.70 RAB9A (0.37) KMT2A
SCHEMBL1190290 0.69 OTUD7B (0.36) CHRNB2CHRNA4NISCHLTA4H
SCHEMBL31343493 0.68 CYP2A6 (0.35) NISCHLTA4H
SCHEMBL16652167 0.68 LTA4H (0.36) NISCHLTA4HSLC6A2SLC6A4
SCHEMBL19859215 0.67 HPGD (0.37) LTA4HP2RX7
SCHEMBL19859207 0.67 CYSLTR1 (0.38) LTA4HP2RX7KMT2A
SCHEMBL16685041 0.64 CHRNB2 (0.40) CHRNB2CHRNA4JAK2HTR1ASLC6A2
SCHEMBL31477187 0.63 GRIN2D (0.32) NISCH
SCHEMBL17633645 0.62 KMT2A (0.40) CHRNB2CHRNA4HTR1AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013050341-A1 AZABENZOXAZINE DERIVATIVES AS CRAC MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2013-04-11 WO disclosed