SCHEMBL14845191

SCHEMBL14845191

Cc1sc(-c2ccccn2)nc1-c1cnc2c(c1)NCC(c1c(F)cccc1F)O2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.37
KMT2A Q03164 4/20 0.37
MAPT P10636 2/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
RECQL P46063 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CYP1A1 P04798 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP1B1 Q16678 1/20 0.33
APEX1 P27695 1/20 0.32
KDM4E B2RXH2 6/20 0.32
GFER P55789 1/20 0.32
ALDH1A1 P00352 4/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
NPC1 O15118 2/20 0.32
TP53 P04637 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14844358 0.75 KDM4E (0.36) RAB9AKMT2AMAPTLMNAGAA
SCHEMBL14841053 0.75 KMT2A (0.36) RAB9AKMT2AMAPTLMNAGAA
SCHEMBL14844536 0.72 CHRNB2 (0.32)
SCHEMBL14840852 0.72 RAB9A (0.35) RAB9AKMT2AMAPTLMNAGAA
SCHEMBL14844199 0.70 CHRNB2 (0.36) KMT2A
SCHEMBL14841201 0.69 APEX1 (0.36) RAB9AKMT2AMAPTLMNAGAA
SCHEMBL14844390 0.66 STIM1 (0.36)
SCHEMBL14844465 0.66 CYP2E1 (0.37) IDO1
SCHEMBL2851161 0.64 KMT2A (0.52) RAB9AKMT2AMAPTLMNAGAA
SCHEMBL14840394 0.64 HTT (0.34) MAPTRECQLCYP1A1CYP1A2CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013050341-A1 AZABENZOXAZINE DERIVATIVES AS CRAC MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2013-04-11 WO disclosed