SCHEMBL14844465

SCHEMBL14844465

CCn1nc(-c2cccnc2)cc1-c1cnc2c(c1)NCC(c1c(F)cccc1F)O2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2E1 P05181 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2A6 P11509 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2B6 P20813 1/20 0.37
CYP2C19 P33261 1/20 0.37
MET P08581 3/20 0.33
CYP11B2 P19099 2/20 0.32
CYP11B1 P15538 1/20 0.32
TBXAS1 P24557 1/20 0.32
F2 P00734 1/20 0.32
HTR2C P28335 3/20 0.32
FYN P06241 1/20 0.31
GUCY1B2 O75343 1/20 0.31
GUCY1A2 P33402 1/20 0.31
GUCY1A1 Q02108 1/20 0.31
GUCY1B1 Q02153 1/20 0.31
LOXL2 Q9Y4K0 1/20 0.31
PGR P06401 1/20 0.31
NR3C2 P08235 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14844261 0.90 HTR2C (0.31) HTR2C
SCHEMBL14844390 0.84 STIM1 (0.36) NR3C2
SCHEMBL14841206 0.76 CYP2E1 (0.37) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL14844358 0.76 KDM4E (0.36) CYP3A4CYP2C19CYP11B2CYP11B1
SCHEMBL14840761 0.73 CYP11B1 (0.37) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL15020516 0.73 ORAI1 (0.41) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL1459710 0.68 CYP19A1 (0.41) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL14844199 0.67 CHRNB2 (0.36)
SCHEMBL14841566 0.66 ALOX5AP (0.32) HTR2C
SCHEMBL14845191 0.66 RAB9A (0.37) IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013050341-A1 AZABENZOXAZINE DERIVATIVES AS CRAC MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2013-04-11 WO disclosed