SCHEMBL14856435

SCHEMBL14856435

CC(=O)Nc1ncc(OC(=O)NC2(C(=O)NCc3ccc(Nc4ccc(F)cc4C(F)(F)F)cn3)CC2)s1

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OGA O60502 6/20 0.33
AURKA O14965 1/20 0.32
CCNE1 P24864 1/20 0.32
CDK2 P24941 1/20 0.32
GRK2 P25098 1/20 0.32
CDK3 Q00526 1/20 0.32
CYP3A4 P08684 1/20 0.32
PIK3CA P42336 1/20 0.32
TRPA1 O75762 2/20 0.32
FAAH O00519 1/20 0.31
P2RX7 Q99572 2/20 0.31
HSD17B10 Q99714 1/20 0.31
RORC P51449 1/20 0.30
CNR2 P34972 1/20 0.30
TRPV1 Q8NER1 1/20 0.30
AR P10275 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14856796 0.89 TRPA1 (0.33) TRPA1FAAHP2RX7RORCCNR2
SCHEMBL2813235 0.89 OGA (0.34) OGAAURKATRPA1P2RX7CNR2
SCHEMBL14856424 0.89 P2RX7 (0.33) AURKATRPA1FAAHP2RX7RORC
SCHEMBL186462 0.83 BACE1 (0.32) TRPA1FAAHP2RX7CNR2TRPV1
SCHEMBL14856710 0.83 FAAH (0.35) TRPA1FAAHP2RX7RORCCNR2
SCHEMBL14856774 0.83 FAAH (0.34) TRPA1FAAHP2RX7TRPV1
SCHEMBL14856577 0.82 FAAH (0.34) TRPA1FAAHP2RX7CNR2TRPV1
SCHEMBL14963913 0.82 HDAC3 (0.40) AURKATRPA1P2RX7CNR2
SCHEMBL2812751 0.82 P2RX7 (0.37) AURKATRPA1P2RX7RORCCNR2
SCHEMBL14856622 0.81 P2RX7 (0.32) AURKATRPA1FAAHP2RX7CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed