SCHEMBL1488884

SCHEMBL1488884

C=CCOc1ccc(C#N)cc1C(F)(F)F

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 2/20 0.50
SSTR4 P31391 1/20 0.45
TRPV4 Q9HBA0 1/20 0.42
SCN9A Q15858 3/20 0.39
ESRRB O95718 1/20 0.39
ESR1 P03372 1/20 0.39
ESRRA P11474 1/20 0.39
ESRRG P62508 1/20 0.39
ESR2 Q92731 1/20 0.39
CTSS P25774 3/20 0.38
AAK1 Q2M2I8 1/20 0.38
KIF11 P52732 1/20 0.38
AGER Q15109 1/20 0.38
PTGDR2 Q9Y5Y4 3/20 0.37
CTSK P43235 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10088897 0.80 CTSS (0.55) MRGPRX4SSTR4TRPV4SCN9ACTSS
SCHEMBL506595 0.77 ALDH1A1 (0.42) ESRRAPTGDR2
SCHEMBL23578526 0.77 MRGPRX4 (0.50) MRGPRX4SSTR4TRPV4SCN9ACTSS
SCHEMBL3496978 0.77 XDH (0.52) MRGPRX4SSTR4TRPV4SCN9AESRRB
SCHEMBL22140450 0.77 TRPV4 (0.43) SSTR4TRPV4KIF11
SCHEMBL6248816 0.75 MRGPRX4 (0.55) MRGPRX4SSTR4TRPV4SCN9ACTSS
SCHEMBL21728097 0.75 AR (0.44) MRGPRX4TRPV4PTGDR2
SCHEMBL28857557 0.75 HPGD (0.40) TRPV4PTGDR2
SCHEMBL22731288 0.74 TRPV4 (0.49) MRGPRX4SSTR4TRPV4SCN9AESRRB
SCHEMBL523319 0.74 ESRRB (0.51) MRGPRX4TRPV4ESRRBESR1ESRRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011035900-A1 NEW THIADIAZOLE DERIVATIVES ALMIRALL, S.A. (ES) 2011-03-31 WO disclosed
WO-2011035900-A1 NEW THIADIAZOLE DERIVATIVES ALMIRALL, S.A. (ES) 2011-03-31 WO disclosed