SCHEMBL1491024

SCHEMBL1491024

C=CC(=O)C=C(c1ccc(C(F)(F)F)cc1)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.52
CES1 P23141 2/20 0.52
GSK3B P49841 2/20 0.49
NR4A1 P22736 1/20 0.49
NR4A2 P43354 1/20 0.49
NR4A3 Q92570 1/20 0.49
TGM2 P21980 1/20 0.49
SRD5A2 P31213 1/20 0.46
PTPN1 P18031 2/20 0.44
CYP1A2 P05177 1/20 0.44
TEAD1 P28347 1/20 0.42
CYP1A1 P04798 4/20 0.41
CYP1B1 Q16678 4/20 0.41
MAOB P27338 1/20 0.41
P4HB P07237 1/20 0.41
MEN1 O00255 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
KMT2A Q03164 1/20 0.40
MMP1 P03956 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1490975 0.78 EPHX2 (0.44) TEAD1TSHRKMT2ATRPV1
SCHEMBL3945570 0.78 NR4A1 (0.61) CES2CES1GSK3BNR4A1NR4A2
SCHEMBL1350180 0.77 CES2 (0.59) CES2CES1GSK3BNR4A1NR4A2
SCHEMBL1490921 0.76 P4HB (0.43) MAOBP4HB
SCHEMBL3945957 0.75 NR4A1 (0.62) CES2CES1GSK3BNR4A1NR4A2
SCHEMBL3945969 0.75 NR4A1 (0.62) CES2CES1GSK3BNR4A1NR4A2
SCHEMBL16502 0.75 AKT1 (0.56) CES2CES1TGM2CYP1A2MEN1
SCHEMBL7934173 0.73 PTPN1 (0.59) CES2CES1GSK3BNR4A1NR4A2
SCHEMBL25252302 0.72 NR4A1 (0.58) CES2CES1GSK3BNR4A1NR4A2
SCHEMBL3944247 0.72 NR4A1 (0.68) CES2CES1GSK3BNR4A1NR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2477698-A2 COMPOUNDS USEFUL AGAINST KINETOPLASTIDEAE PARASITES Centre National de la Recherche Scientifique (FR) 2012-07-25 EP disclosed
WO-2011033115-A2 COMPOUNDS USEFUL AGAINST KINETOPLASTIDEAE PARASITES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2011-03-24 WO disclosed