SCHEMBL1490975

SCHEMBL1490975

C=CC(=O)C=C(c1ccc(OC(F)(F)F)cc1)c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 3/20 0.44
TRPV1 Q8NER1 3/20 0.43
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
FAAH O00519 1/20 0.41
HRH3 Q9Y5N1 2/20 0.40
KMT2A Q03164 1/20 0.40
GAA P10253 1/20 0.40
TEAD1 P28347 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
AURKA O14965 1/20 0.39
TPX2 Q9ULW0 1/20 0.39
TLR7 Q9NYK1 1/20 0.39
NR1H4 Q96RI1 1/20 0.39
MTOR P42345 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16563109 0.80 ALDH5A1 (0.52) EPHX2TRPV1NPC1RAB9AFAAH
SCHEMBL1490910 0.78 CES2 (0.52) RAB9AALDH1A1HSD17B10
SCHEMBL1491024 0.78 CES2 (0.52) TRPV1KMT2ATEAD1TSHR
SCHEMBL1490630 0.78 APP (0.46) RAB9AKMT2A
SCHEMBL11773412 0.75 MMP2 (0.47) EPHX2TRPV1NPC1RAB9AFAAH
SCHEMBL23930173 0.75 HSD11B1 (0.46) EPHX2TRPV1NPC1RAB9AFAAH
SCHEMBL23930171 0.75 HSD11B1 (0.46) EPHX2TRPV1NPC1RAB9AFAAH
SCHEMBL7786865 0.75 CA1 (0.50) RAB9AKMT2AGAAALDH1A1TSHR
SCHEMBL28186415 0.74 EPHX2 (0.50) EPHX2TRPV1NPC1RAB9AFAAH
SCHEMBL514074 0.73 EPHX2 (0.53) EPHX2TRPV1NPC1RAB9AFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2477698-A2 COMPOUNDS USEFUL AGAINST KINETOPLASTIDEAE PARASITES Centre National de la Recherche Scientifique (FR) 2012-07-25 EP disclosed
WO-2011033115-A2 COMPOUNDS USEFUL AGAINST KINETOPLASTIDEAE PARASITES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2011-03-24 WO disclosed