SCHEMBL1491306

SCHEMBL1491306

CC(=O)c1ccc(S(=O)(=O)O)c2ccncc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HASPIN Q8TF76 1/20 0.37
COMT P21964 1/20 0.36
NAPRT Q6XQN6 1/20 0.35
CYP1A2 P05177 2/20 0.34
KDM4E B2RXH2 1/20 0.34
HTT P42858 1/20 0.34
ALDH1A1 P00352 1/20 0.34
ALOX15 P16050 1/20 0.34
HIF1A Q16665 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TTR P02766 1/20 0.33
SIRT3 Q9NTG7 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
BRAF P15056 1/20 0.33
CSNK1A1 P48729 1/20 0.33
CSNK1D P48730 1/20 0.33
CSNK1E P49674 1/20 0.33
CSNK1G2 P78368 1/20 0.33
CSNK1G1 Q9HCP0 1/20 0.33
TET2 Q6N021 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20836182 0.83 NAPRT (0.44) COMTNAPRTCYP1A2KDM4EALDH1A1
SCHEMBL30842108 0.83 NAPRT (0.44) COMTNAPRTCYP1A2KDM4EALDH1A1
SCHEMBL8031733 0.81 NAPRT (0.42) COMTNAPRTCYP1A2KDM4EHTT
SCHEMBL1491302 0.79 POLB (0.38) COMTNAPRTCYP1A2ALDH1A1ALOX15
SCHEMBL4349196 0.78 TTR (0.46) COMTCYP1A2KDM4EALDH1A1ALOX15
SCHEMBL16508198 0.78 CASP6 (0.44) KDM4EALDH1A1BRAFCA1CA2
SCHEMBL16508188 0.76 EP300 (0.56) COMTNAPRTCYP1A2KDM4EHTT
SCHEMBL21801051 0.73 KDM4E (0.53) KDM4EHTTALDH1A1HSD17B10
SCHEMBL1491313 0.73 ROCK2 (0.61) CYP1A2KDM4EHTTALDH1A1HIF1A
SCHEMBL16508210 0.73 HASPIN (0.44) HASPINNAPRTKDM4EHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2296472-A1 COMPOUNDS FOR RHO KINASE INHIBITION AND FOR IMPROVING LEARNING AND MEMORY Amnestix, Inc. (US) 2011-03-23 EP disclosed
WO-2009151845-A9 COMPOUNDS FOR RHO KINASE INHIBITION AND FOR IMPROVING LEARNING AND MEMORY AMNESTIX, INC. (US) 2010-01-28 WO disclosed
WO-2009151845-A1 COMPOUNDS FOR RHO KINASE INHIBITION AND FOR IMPROVING LEARNING AND MEMORY AMNESTIX, INC. (US) 2009-12-17 WO disclosed