SCHEMBL14919176

SCHEMBL14919176

COc1ccc(NC(=O)C(C)(C)CCCCc2noc(C(F)(F)F)n2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.45
PDK2 Q15119 1/20 0.45
PDK3 Q15120 1/20 0.45
PDK4 Q16654 1/20 0.45
SMN1; SMN2 Q16637 4/20 0.43
MAPT P10636 3/20 0.43
TP53 P04637 2/20 0.43
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
TDP1 Q9NUW8 1/20 0.38
RAF1 P04049 1/20 0.38
HDAC1 Q13547 3/20 0.38
HDAC8 Q9BY41 3/20 0.38
HDAC2 Q92769 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KDM4E B2RXH2 1/20 0.38
CYP3A4 P08684 1/20 0.38
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14918896 0.89 MEN1 (0.41) SMN1; SMN2MAPTNPC1RAB9AMEN1
SCHEMBL14918924 0.89 HDAC1 (0.48) PDK1PDK2PDK3PDK4SMN1; SMN2
SCHEMBL14918747 0.87 HDAC6 (0.48) MAPTMEN1KMT2AHDAC1HDAC8
SCHEMBL14918889 0.86 MEN1 (0.38) SMN1; SMN2MAPTTP53MEN1KMT2A
SCHEMBL14919184 0.85 L3MBTL1 (0.57) SMN1; SMN2MAPTTP53NPC1RAB9A
SCHEMBL14918545 0.84 L3MBTL1 (0.56) SMN1; SMN2MAPTTP53MEN1KMT2A
SCHEMBL14918539 0.84 L3MBTL1 (0.56) SMN1; SMN2MAPTTP53MEN1KMT2A
SCHEMBL14918439 0.84 L3MBTL1 (0.56) SMN1; SMN2MAPTTP53MEN1KMT2A
SCHEMBL14919092 0.83 L3MBTL1 (0.55) SMN1; SMN2MAPTTP53NPC1RAB9A
SCHEMBL14918730 0.82 HDAC6 (0.40) HDAC1HDAC8LMNAHTTHDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013066836-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2013-05-10 WO claimed