SCHEMBL14939855

SCHEMBL14939855

O=C1c2ccccc2C(=O)C1(c1ccc2ccccc2n1)N1CCN(Cc2ccccc2)CC1

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.65
GRIN2B Q13224 1/20 0.47
KMT2A Q03164 1/20 0.44
SIGMAR1 Q99720 3/20 0.43
MMP2 P08253 1/20 0.42
MMP9 P14780 1/20 0.42
DRD2 P14416 2/20 0.42
HTR2A P28223 2/20 0.42
HTR2C P28335 2/20 0.42
HTR2B P41595 2/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
ADAM17 P78536 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14940076 0.85 NPSR1 (0.46) NPSR1GRIN2BKMT2ALMNAMAPT
SCHEMBL14939887 0.85 NPSR1 (0.64) NPSR1SIGMAR1MMP2MMP9DRD2
SCHEMBL14940429 0.84 NPSR1 (0.46) NPSR1GRIN2BKMT2AKDM4EALDH1A1
SCHEMBL14939501 0.84 HTR1A (0.49) NPSR1SIGMAR1DRD2HTR2BKDM4E
SCHEMBL14940072 0.83 L3MBTL1 (0.52) NPSR1KMT2ADRD2HTR2BKDM4E
SCHEMBL14939426 0.82 NPSR1 (0.67) NPSR1KMT2ASIGMAR1MMP2MMP9
SCHEMBL14940084 0.82 MEN1 (0.47) NPSR1KMT2ADRD2HTR2BKDM4E
SCHEMBL14939341 0.81 NPSR1 (0.65) NPSR1KMT2ASIGMAR1MMP2MMP9
SCHEMBL14939259 0.81 NPSR1 (0.65) NPSR1SIGMAR1MMP2MMP9DRD2
SCHEMBL14939647 0.80 NPSR1 (0.74) NPSR1KMT2ASIGMAR1MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed