SCHEMBL14943017

SCHEMBL14943017

CCCOc1ccc2sc(S(=O)(=O)NCP(=O)(O)Oc3ccc(C#N)nc3)cc2c1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 2/20 0.34
LMNA P02545 1/20 0.34
KAT6A Q92794 2/20 0.34
CA2 P00918 3/20 0.33
SCD O00767 1/20 0.33
LRRK2 Q5S007 1/20 0.32
FBP1 P09467 1/20 0.32
SLC40A1 Q9NP59 1/20 0.31
ACACB O00763 2/20 0.31
S1PR1 P21453 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13032085 0.92 CA2 (0.33) CA2SLC40A1
SCHEMBL14943016 0.87 LMNA (0.35) CLK1LMNAKAT6ACA2SCD
SCHEMBL14943032 0.84 TRPV4 (0.37) KAT6A
SCHEMBL14942987 0.83 CA2 (0.31) CA2
SCHEMBL14943013 0.82 AR (0.36) CLK1
SCHEMBL13032088 0.80 CA2 (0.35) CA2FBP1
SCHEMBL13032075 0.78 TRPV4 (0.39)
SCHEMBL14931181 0.77 TRPV4 (0.37)
SCHEMBL3483772 0.77 TRPV4 (0.36)
SCHEMBL14931498 0.77 TRPV4 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8440643-B2 Inhibitors of beta-lactamase METHYLGENE INC. (CA) 2013-05-14 US disclosed