SCHEMBL14955294

SCHEMBL14955294

O=c1[nH]nccc1-c1cccnc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.58
CYP2E1 P05181 1/20 0.58
CYP2B6 P20813 1/20 0.58
HPGDS O60760 1/20 0.51
BTK Q06187 1/20 0.49
ALDH1A1 P00352 3/20 0.48
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
METAP2 P50579 1/20 0.47
SIRT3 Q9NTG7 1/20 0.47
P4HTM Q9NXG6 1/20 0.46
NUDT1 P36639 1/20 0.45
VHL P40337 1/20 0.44
AURKA O14965 1/20 0.44
TTK P33981 1/20 0.44
AURKB Q96GD4 1/20 0.44
INCENP Q9NQS7 1/20 0.44
ALK Q9UM73 1/20 0.44
PIM1 P11309 2/20 0.43
PIM3 Q86V86 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL918364 0.81 SCN4A (0.52) HPGDSBTKALDH1A1CYP1A2METAP2
Hydrochloric Acid SCHEMBL30014721 0.79 SCN4A (0.50) HPGDSBTKALDH1A1CYP1A2METAP2
SCHEMBL8213047 0.79 HPGDS (0.53) CYP2A6CYP2E1CYP2B6HPGDSBTK
SCHEMBL4787445 0.78 SCN4A (0.48) HPGDSALDH1A1AURKAPIM1GSK3B
SCHEMBL11094847 0.77 PDPK1 (0.52) ALDH1A1CYP1A2CYP3A4AURKATTK
SCHEMBL1456892 0.76 HCAR2 (0.41) ALDH1A1PIM1LMNAHSD17B10
SCHEMBL2101504 0.75 NUDT1 (0.49) CYP2A6CYP2E1CYP2B6BTKALDH1A1
SCHEMBL31235677 0.75 NUDT1 (0.49) CYP2A6CYP2E1CYP2B6BTKALDH1A1
SCHEMBL28815828 0.74 RPS6KA3 (0.47) PIM1GSK3B
SCHEMBL28051817 0.74 NOTUM (0.62) NUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119998271-A Pyridone compound and preparation method and application thereof 深圳信立泰药业股份有限公司 2025-05-13 CN disclosed
US-9221806-B2 2-(heterocyclylbenzyl)pyridazinone derivatives MERCK PATENT GMBH (DE) 2015-12-29 US disclosed
US-20130131037-A1 2-(HETEROCYCLYLBENZYL)PYRIDAZINONE DERIVATIVES MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 2013-05-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130131037-A1 2-(HETEROCYCLYLBENZYL)PYRIDAZINONE DERIVATIVES RET, MET, ERBB2 CYP2A6 1525/4885CYP2E1 1028/4885CYP2B6 710/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.