SCHEMBL14966243

SCHEMBL14966243

CN(C)C(=O)c1cccc(-c2ccc(CN3CCOc4nc([N+](=O)[O-])cn4CC3)cc2)c1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TNIK Q9UKE5 1/20 0.45
AXL P30530 1/20 0.40
MERTK Q12866 1/20 0.40
ERN1 O75460 1/20 0.39
FAAH O00519 1/20 0.38
MGLL Q99685 1/20 0.38
ADORA2A P29274 1/20 0.38
DRD2 P14416 1/20 0.38
ALDH1A1 P00352 3/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
ACHE P22303 1/20 0.37
CHEK1 O14757 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
SUCNR1 Q9BXA5 1/20 0.36
DAGLA Q9Y4D2 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965511 0.90 LTA4H (0.40) FAAHALDH1A1LMNAMAPTMEN1
SCHEMBL14965626 0.90 LTA4H (0.40) FAAHALDH1A1LMNAMAPTMEN1
SCHEMBL14965560 0.89 HIF1A (0.40) DRD2ALDH1A1LMNAMAPTCHEK1
SCHEMBL14971109 0.87 TP53 (0.40) ALDH1A1LMNAMAPT
SCHEMBL14965896 0.87 SUCNR1 (0.40) TNIKALDH1A1LMNAMAPTMEN1
SCHEMBL14969471 0.86 KDM4E (0.41) TNIKERN1ALDH1A1LMNAMAPT
SCHEMBL14965684 0.86 CHKA (0.45) ERN1FAAHMGLLALDH1A1LMNA
SCHEMBL14965672 0.85 DRD4 (0.47) DRD2ALDH1A1ACHEMEN1KMT2A
SCHEMBL14971108 0.84 ALDH1A1 (0.44) FAAHMGLLALDH1A1LMNAMAPT
SCHEMBL14965746 0.84 DRD2 (0.41) DRD2ALDH1A1LMNAMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed