SCHEMBL14965673

SCHEMBL14965673

N#Cc1ccc(-c2ccc(CN3CCOc4nc([N+](=O)[O-])cn4CC3)nc2)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.36
HSD11B1 P28845 1/20 0.34
SRC P12931 1/20 0.34
KCNH2 Q12809 4/20 0.34
KCNJ1 P48048 1/20 0.34
HRH3 Q9Y5N1 2/20 0.33
GPR39 O43194 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
HRH2 P25021 1/20 0.33
HRH1 P35367 1/20 0.33
CHEK1 O14757 1/20 0.33
ACHE P22303 1/20 0.33
TNIK Q9UKE5 1/20 0.32
MAPT P10636 1/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
CYP11B1 P15538 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965986 0.88 KCNJ1 (0.41) KCNH2KCNJ1HRH3MAPTALDH1A1
SCHEMBL14965894 0.86 HIF1A (0.41) MCHR1KCNH2TNIK
SCHEMBL14965893 0.85 SCN9A (0.37) MCHR1HSD11B1SRCKCNH2KCNJ1
SCHEMBL14965790 0.84 DRD2 (0.38) SRCKCNH2KCNJ1TNIKCYP11B1
SCHEMBL14966215 0.84 CYP11B1 (0.43) HSD11B1SRCKCNH2KCNJ1HRH3
SCHEMBL14965795 0.83 CYP11B1 (0.45) MCHR1SRCKCNH2KCNJ1CYP11B1
SCHEMBL14965410 0.83 DRD2 (0.38) SRCKCNH2KDM4EALDH1A1
SCHEMBL14965939 0.82 PDE9A (0.39) SRCKCNH2KCNJ1KDM4EALDH1A1
SCHEMBL14965663 0.82 KCNH2 (0.35) KCNH2KCNJ1HRH3MAPTKDM4E
SCHEMBL14965508 0.82 CAMKK2 (0.37) SRCKCNH2KCNJ1HRH3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed