SCHEMBL14965663

SCHEMBL14965663

O=[N+]([O-])c1cn2c(n1)OCCN(Cc1ccc(Br)cn1)CC2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.35
ALDH1A1 P00352 4/20 0.34
KDM4E B2RXH2 2/20 0.34
LMNA P02545 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
MAPT P10636 2/20 0.33
CHRM1 P11229 1/20 0.33
PDE2A O00408 1/20 0.33
TSHR P16473 1/20 0.32
HRH3 Q9Y5N1 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
KCNJ1 P48048 1/20 0.31
DRD4 P21917 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
POLB P06746 2/20 0.31
MAPK1 P28482 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965999 0.85 ALDH1A1 (0.43) ALDH1A1KDM4ELMNAMAPTCHRM1
SCHEMBL14965813 0.83 ALDH1A1 (0.53) ALDH1A1KDM4ELMNACYP1A2CYP2C19
SCHEMBL14965974 0.82 FAAH (0.41) KCNH2ALDH1A1KDM4ELMNAMAPT
SCHEMBL14965894 0.82 HIF1A (0.41) KCNH2CHRM1
SCHEMBL14965673 0.82 MCHR1 (0.36) KCNH2ALDH1A1KDM4ECYP1A2CYP2C19
SCHEMBL14966128 0.82 ALDH1A1 (0.38) KCNH2ALDH1A1LMNAMAPTCHRM1
SCHEMBL14965410 0.81 DRD2 (0.38) KCNH2ALDH1A1KDM4EDRD4POLB
SCHEMBL14965821 0.80 ALDH1A1 (0.33) KCNH2ALDH1A1KDM4ELMNAMAPT
SCHEMBL14965699 0.80 SMN1; SMN2 (0.43) ALDH1A1KDM4ELMNAMAPTSMN1; SMN2
SCHEMBL14965623 0.79 CYP2A13 (0.48) ALDH1A1KDM4ELMNATSHRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed