SCHEMBL14965706

SCHEMBL14965706

O=C(c1ccc(Oc2ccc(Br)cc2)cc1)N1CCOc2nc([N+](=O)[O-])cn2CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
POLB P06746 2/20 0.45
ALDH1A1 P00352 2/20 0.44
MAPT P10636 2/20 0.44
HSP90AA1 P07900 1/20 0.44
GAA P10253 1/20 0.44
MAPK1 P28482 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
HPGD P15428 3/20 0.42
LMNA P02545 2/20 0.42
RAB9A P51151 1/20 0.42
TSHR P16473 1/20 0.39
NAAA Q02083 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965651 0.94 HPGD (0.43) KMT2APOLBALDH1A1MAPTHSP90AA1
SCHEMBL14965598 0.91 NAAA (0.49) MEN1KMT2APOLBALDH1A1MAPT
SCHEMBL14965860 0.82 ALDH1A1 (0.52) MEN1KMT2AALDH1A1MAPTGAA
SCHEMBL14965827 0.81 NAAA (0.53) KMT2AALDH1A1MAPTGAAMAPK1
SCHEMBL14966196 0.81 ALDH1A1 (0.49) MEN1KMT2APOLBALDH1A1MAPT
SCHEMBL14965625 0.80 SMN1; SMN2 (0.40) POLBALDH1A1MAPTGAASMN1; SMN2
SCHEMBL14965900 0.78 GPR183 (0.41) MEN1KMT2APOLBALDH1A1MAPT
SCHEMBL14965793 0.76 HPGD (0.53) MEN1KMT2AALDH1A1MAPTGAA
SCHEMBL14965608 0.75 CHRM1 (0.48) KCNH2
SCHEMBL14966002 0.75 HPGD (0.54) MEN1KMT2AALDH1A1SMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed