SCHEMBL14965860

SCHEMBL14965860

O=C(c1cccc(Br)c1)N1CCOc2nc([N+](=O)[O-])cn2CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.52
TP53 P04637 1/20 0.52
HPGD P15428 1/20 0.47
KDM4E B2RXH2 1/20 0.47
MAPT P10636 2/20 0.46
GAA P10253 1/20 0.46
MAPK1 P28482 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
KMT2A Q03164 3/20 0.45
MEN1 O00255 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA7 P43166 1/20 0.45
CA9 Q16790 1/20 0.45
CA14 Q9ULX7 1/20 0.45
RXFP1 Q9HBX9 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965651 0.88 HPGD (0.43) ALDH1A1HPGDKDM4EMAPTGAA
SCHEMBL14966196 0.85 ALDH1A1 (0.49) ALDH1A1HPGDKDM4EMAPTGAA
SCHEMBL14965706 0.82 MEN1 (0.45) ALDH1A1HPGDMAPTGAAMAPK1
SCHEMBL14965998 0.82 CYP11B2 (0.45) HPGDKDM4EKMT2AMEN1RAB9A
SCHEMBL14965625 0.80 SMN1; SMN2 (0.40) ALDH1A1HPGDKDM4EMAPTGAA
SCHEMBL14965888 0.80 PIK3CA (0.43) ALDH1A1KDM4EMAPTGAAMAPK1
SCHEMBL14965598 0.79 NAAA (0.49) ALDH1A1HPGDKDM4EMAPTGAA
SCHEMBL14965699 0.77 SMN1; SMN2 (0.43) ALDH1A1KDM4EMAPTMAPK1TDP1
SCHEMBL14971106 0.77 POLB (0.56) KMT2AMEN1SMN1; SMN2CA12CA1
SCHEMBL14965869 0.76 ALDH1A1 (0.41) ALDH1A1MAPTGAAKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed