SCHEMBL14965723

SCHEMBL14965723

N#Cc1ccc(N2CCN(c3nccc(N4CCOc5nc([N+](=O)[O-])cn5CC4)n3)CC2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.39
SLC6A9 P48067 1/20 0.37
SLC6A5 Q9Y345 1/20 0.37
POLB P06746 1/20 0.37
JAK2 O60674 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
GAA P10253 1/20 0.35
ALDH1A1 P00352 2/20 0.33
KDR P35968 1/20 0.33
USP30 Q70CQ3 1/20 0.33
SUV39H2 Q9H5I1 2/20 0.33
PTGS1 P23219 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
MAPT P10636 1/20 0.33
KDM4E B2RXH2 1/20 0.32
TP53 P04637 1/20 0.32
CTSL P07711 1/20 0.32
CTSB P07858 1/20 0.32
CTSS P25774 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965984 0.88 MAPT (0.42) POLBL3MBTL1ALDH1A1SUV39H2MAPT
SCHEMBL14965789 0.88 CYP1A2 (0.40) POLBGAAALDH1A1USP30SUV39H2
SCHEMBL14965943 0.86 GBA1 (0.40) POLBGAAALDH1A1MAPTKDM4E
SCHEMBL14965857 0.82 ENPP2 (0.36) POLBGAAALDH1A1SUV39H2SLC6A2
SCHEMBL14971157 0.81 PIK3CA (0.43) L3MBTL1GAAALDH1A1MAPTKDM4E
SCHEMBL14965923 0.81 OGA (0.46) SLC6A2
SCHEMBL14965774 0.80 GBA1 (0.32) POLBL3MBTL1ALDH1A1MAPT
SCHEMBL14965617 0.78 TRPV1 (0.45) POLBALDH1A1
SCHEMBL14966123 0.77 KMT2A (0.52) SLC6A9SLC6A5POLBALDH1A1MAPT
SCHEMBL14966084 0.75 SLC6A9 (0.41) SLC6A9SLC6A5JAK2ALDH1A1PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed