SCHEMBL14965857

SCHEMBL14965857

O=[N+]([O-])c1cn2c(n1)OCCN(c1ccnc(N3CCN(c4cccc(F)c4)CC3)n1)CC2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 2/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
MAPT P10636 4/20 0.35
ALDH1A1 P00352 2/20 0.35
SUV39H2 Q9H5I1 2/20 0.34
PIK3CD O00329 2/20 0.34
SCN9A Q15858 1/20 0.34
TRPV1 Q8NER1 1/20 0.33
PIK3R1 P27986 1/20 0.33
LMNA P02545 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
GAA P10253 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
POLB P06746 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965984 0.89 MAPT (0.42) MEN1KMT2AMAPTALDH1A1SUV39H2
SCHEMBL14965789 0.85 CYP1A2 (0.40) KMT2AMAPTALDH1A1SUV39H2PIK3CD
SCHEMBL14965943 0.85 GBA1 (0.40) MEN1KMT2AMAPTALDH1A1LMNA
SCHEMBL14965723 0.82 AOC3 (0.39) MAPTALDH1A1SUV39H2SCN9AGAA
SCHEMBL14965774 0.81 GBA1 (0.32) MAPTALDH1A1PIK3CDTRPV1LMNA
SCHEMBL14965617 0.77 TRPV1 (0.45) ALDH1A1TRPV1CYP1A2CYP2C9POLB
SCHEMBL14971157 0.77 PIK3CA (0.43) MEN1KMT2AMAPTALDH1A1LMNA
SCHEMBL14965808 0.77 LMNA (0.47) ENPP2MEN1KMT2AMAPTALDH1A1
SCHEMBL14965834 0.73 OGA (0.49) MAPTALDH1A1SLC6A2SLC6A3MAPK1
SCHEMBL14966122 0.72 OGA (0.41) TRPV1SMN1; SMN2SLC6A2SLC6A3MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed