SCHEMBL14965774

SCHEMBL14965774

O=[N+]([O-])c1cn2c(n1)OCCN(c1ccnc(N3CC=CCC3)n1)CC2

nearest known ligand 0.32

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.32
KCNH2 Q12809 3/20 0.31
TRPV1 Q8NER1 1/20 0.31
LMNA P02545 1/20 0.31
CYP1A2 P05177 2/20 0.31
CYP2C9 P11712 2/20 0.31
SORD Q00796 1/20 0.31
POLB P06746 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
NPC1 O15118 1/20 0.30
MAPT P10636 1/20 0.30
RAB9A P51151 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
PIK3CD O00329 1/20 0.30
PIK3CA P42336 1/20 0.30
CHRM1 P11229 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965789 0.87 CYP1A2 (0.40) LMNACYP1A2CYP2C9POLBALDH1A1
SCHEMBL14965943 0.87 GBA1 (0.40) GBA1KCNH2LMNACYP1A2CYP2C9
SCHEMBL14965984 0.86 MAPT (0.42) GBA1LMNACYP1A2CYP2C9SORD
SCHEMBL14965857 0.81 ENPP2 (0.36) TRPV1LMNACYP1A2CYP2C9POLB
SCHEMBL14965617 0.81 TRPV1 (0.45) KCNH2TRPV1CYP1A2CYP2C9SORD
SCHEMBL14965723 0.80 AOC3 (0.39) POLBALDH1A1MAPTL3MBTL1
SCHEMBL14965834 0.76 OGA (0.49) ALDH1A1MAPTL3MBTL1
SCHEMBL14971157 0.76 PIK3CA (0.43) LMNAALDH1A1HPGDMAPTL3MBTL1
SCHEMBL14965871 0.75 ALDH1A1 (0.42) LMNAPOLBALDH1A1MAPTL3MBTL1
SCHEMBL14965636 0.72 HRH4 (0.47) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed