SCHEMBL14965907

SCHEMBL14965907

COc1ncccc1-c1ccc(CN2CCOc3nc([N+](=O)[O-])cn3CC2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 3/20 0.37
NAAA Q02083 1/20 0.37
CHRM1 P11229 1/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
GSK3B P49841 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PIK3CA P42336 1/20 0.35
ALDH1A1 P00352 2/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
KCNJ1 P48048 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TSHR P16473 1/20 0.34
DRD2 P14416 1/20 0.34
DRD4 P21917 1/20 0.34
DRD3 P35462 1/20 0.34
CTSB P07858 1/20 0.34
KCNH2 Q12809 3/20 0.34
ABCB1 P08183 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965823 0.87 CLK2 (0.39) CHRM1L3MBTL1ALDH1A1LMNAMAPT
SCHEMBL14966106 0.84 SMN1; SMN2 (0.46) CHRM1ALDH1A1LMNAMAPTKCNJ1
SCHEMBL14965775 0.83 L3MBTL1 (0.41) CHRM1GSK3BL3MBTL1ALDH1A1LMNA
SCHEMBL14965513 0.83 LSS (0.46) CHRM1ALDH1A1LMNAMAPTKCNJ1
SCHEMBL14965703 0.83 SMN1; SMN2 (0.49) CHRM1ALDH1A1LMNAMAPTKCNJ1
SCHEMBL14965825 0.82 CD274 (0.38) CHRM1PIK3CAALDH1A1LMNAMAPT
SCHEMBL14965541 0.82 CD274 (0.39) TBK1CHRM1PIK3CAALDH1A1LMNA
SCHEMBL14971108 0.82 ALDH1A1 (0.44) L3MBTL1ALDH1A1LMNAMAPTKCNJ1
SCHEMBL14966132 0.81 DRD4 (0.44) ALDH1A1LMNAMAPTSMN1; SMN2DRD2
SCHEMBL14965550 0.81 SLC2A1 (0.39) ALDH1A1LMNAMAPTKCNJ1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed