SCHEMBL14965823

SCHEMBL14965823

O=[N+]([O-])c1cn2c(n1)OCCN(Cc1ccc(-c3cccnc3F)cc1)CC2

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CLK2 P49760 1/20 0.39
CLK3 P49761 1/20 0.39
DYRK1A Q13627 1/20 0.39
CHRM1 P11229 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
KCNJ1 P48048 3/20 0.36
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SOS1 Q07889 1/20 0.36
TSHR P16473 1/20 0.35
KCNH2 Q12809 5/20 0.35
TGFBR1 P36897 2/20 0.34
CACNA1C Q13936 1/20 0.34
SCN5A Q14524 1/20 0.34
CTSB P07858 1/20 0.33
AKT1 P31749 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965907 0.87 TBK1 (0.37) CHRM1L3MBTL1KCNJ1ALDH1A1LMNA
SCHEMBL14965775 0.85 L3MBTL1 (0.41) CHRM1L3MBTL1KCNJ1ALDH1A1KDM4E
SCHEMBL14971108 0.84 ALDH1A1 (0.44) L3MBTL1KCNJ1ALDH1A1KDM4ELMNA
SCHEMBL14965513 0.83 LSS (0.46) DYRK1ACHRM1KCNJ1ALDH1A1LMNA
SCHEMBL14965620 0.83 ALDH1A1 (0.38) CHRM1L3MBTL1KCNJ1ALDH1A1LMNA
SCHEMBL14965550 0.83 SLC2A1 (0.39) DYRK1AKCNJ1ALDH1A1LMNAMAPT
SCHEMBL14965746 0.82 DRD2 (0.41) CHRM1KCNJ1ALDH1A1LMNAMAPT
SCHEMBL14965773 0.81 L3MBTL1 (0.46) L3MBTL1KCNJ1ALDH1A1KDM4ELMNA
SCHEMBL14965750 0.81 CHKA (0.43) CHRM1L3MBTL1KCNJ1ALDH1A1KDM4E
SCHEMBL14965918 0.80 ALDH1A1 (0.37) CHRM1L3MBTL1KCNJ1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed