SCHEMBL14965897

SCHEMBL14965897

O=C(O)c1ccc(-c2cccc(CN3CCOc4nc([N+](=O)[O-])cn4CC3)n2)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
CXCR4 P61073 1/20 0.34
ALDH1A1 P00352 3/20 0.33
ALOX5 P09917 2/20 0.33
PTGES2 Q9H7Z7 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
RARA P10276 1/20 0.32
RARB P10826 1/20 0.32
PTGES O14684 1/20 0.32
EGLN1 Q9GZT9 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965895 1.00 HTR1A (0.35) HTR1ADRD2CXCR4ALDH1A1ALOX5
SCHEMBL14971086 0.88 ALDH1A1 (0.41) ALDH1A1MAPTTSHRMAPK1MEN1
SCHEMBL14965893 0.86 SCN9A (0.37) HTR1ADRD2CXCR4KCNH2HSD11B1
SCHEMBL14966129 0.86 SCN9A (0.37) HTR1ADRD2CXCR4KCNH2SLC2A1
SCHEMBL14965368 0.85 KCNJ1 (0.40) ALDH1A1KDM4EMAPTMAPK1MEN1
SCHEMBL14965407 0.84 KCNJ1 (0.42) ALDH1A1KDM4EMAPTMAPK1MEN1
SCHEMBL14965730 0.83 DRD2 (0.37) HTR1ADRD2CXCR4ALDH1A1KDM4E
SCHEMBL14966317 0.83 LOXL2 (0.42) HTR1ADRD2ALDH1A1MEN1KMT2A
SCHEMBL14966011 0.81 MTOR (0.37) HTR1ADRD2ALDH1A1KCNH2AOC3
SCHEMBL14966353 0.81 JAK2 (0.37) HTR1ADRD2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed