SCHEMBL14966199

SCHEMBL14966199

O=C(O)c1ccc(CCOc2ccncn2)cc1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 3/20 0.45
CYP4A11 Q02928 3/20 0.45
TBXAS1 P24557 3/20 0.42
NAPRT Q6XQN6 1/20 0.42
POLB P06746 1/20 0.40
NR4A2 P43354 1/20 0.40
LTA4H P09960 1/20 0.39
PDE4D Q08499 1/20 0.39
MAPT P10636 1/20 0.39
RARB P10826 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
ALDH1A1 P00352 1/20 0.39
PIM1 P11309 1/20 0.38
PIM2 Q9P1W9 1/20 0.38
PKM P14618 1/20 0.38
GCK P35557 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14967310 0.85 CYP4A11 (0.49) CYP4F2CYP4A11MAPTALDH1A1PKM
SCHEMBL14967550 0.81 POLB (0.55) CYP4F2CYP4A11POLBNR4A2ALDH1A1
SCHEMBL14966872 0.80 LTA4H (0.56) CYP4F2CYP4A11TBXAS1NAPRTPOLB
SCHEMBL14967498 0.78 ELOVL1 (0.40) LTA4HPIM1PIM2
SCHEMBL14967192 0.75 POLB (0.51) CYP4F2CYP4A11TBXAS1POLBNR4A2
SCHEMBL6769826 0.73 NAPRT (0.64) TBXAS1NAPRTPOLBRARBALDH1A1
SCHEMBL4255608 0.73 MAPT (0.59) NR4A2MAPTGCK
Hydrochloric Acid SCHEMBL3896488 0.72 NAPRT (0.61) TBXAS1NAPRTPOLBRARBALDH1A1
SCHEMBL11891840 0.72 SRD5A2 (0.54) NAPRTPOLB
SCHEMBL5390756 0.71 PKM (0.73) NR4A2PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2780014-A1 MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF Constellation Pharmaceuticals, Inc. (US) 2014-09-24 EP disclosed
WO-2013075083-A1 MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF CONSTELLATION PHARMACEUTICALS (US) 2013-05-23 WO disclosed