SCHEMBL14965835

SCHEMBL14965835

O=C(c1ccc(-c2cc(CN3CCOc4nc([N+](=O)[O-])cn4CC3)ccn2)cc1F)N1CCCC1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MTOR P42345 8/20 0.37
JAK2 O60674 2/20 0.35
JAK1 P23458 2/20 0.35
TYK2 P29597 2/20 0.35
JAK3 P52333 2/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
PIK3CA P42336 2/20 0.34
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965806 0.94 MET (0.39) MTORJAK2JAK1TYK2JAK3
SCHEMBL14965820 0.90 JAK2 (0.37) MTORJAK2JAK1TYK2JAK3
SCHEMBL14965666 0.88 LRRK2 (0.36) JAK2JAK1TYK2JAK3
SCHEMBL14965574 0.88 HDAC4 (0.36) PIK3CA
SCHEMBL14966211 0.87 MTOR (0.38) MTORPIK3CA
SCHEMBL14965517 0.86 FGFR1 (0.40) ALDH1A1
SCHEMBL14966353 0.86 JAK2 (0.37) JAK2JAK1TYK2JAK3LMNA
SCHEMBL14966081 0.84 KCNJ1 (0.39) MTORJAK2JAK1TYK2JAK3
SCHEMBL14965844 0.84 LMNA (0.35) JAK2JAK1TYK2JAK3LMNA
SCHEMBL14966238 0.83 MET (0.41) MTORJAK2JAK1TYK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed