SCHEMBL14965666

SCHEMBL14965666

CN(C)C(=O)c1ccc(-c2cc(CN3CCOc4nc([N+](=O)[O-])cn4CC3)ccn2)cc1F

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.36
MET P08581 1/20 0.36
TBK1 Q9UHD2 12/20 0.33
CCNT1 O60563 3/20 0.33
FLT3 P36888 3/20 0.33
CDK9 P50750 3/20 0.33
IKBKE Q14164 3/20 0.33
RPS6KA6 Q9UK32 3/20 0.33
STK17A Q9UEE5 1/20 0.33
JAK2 O60674 3/20 0.33
JAK1 P23458 3/20 0.33
TYK2 P29597 3/20 0.33
JAK3 P52333 3/20 0.33
HTR1A P08908 1/20 0.32
DRD2 P14416 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965652 0.90 GPR119 (0.38) LRRK2METJAK2JAK1TYK2
SCHEMBL14966211 0.88 MTOR (0.38) METTBK1
SCHEMBL14965835 0.88 MTOR (0.37) JAK2JAK1TYK2JAK3
SCHEMBL14965574 0.88 HDAC4 (0.36) METTBK1
SCHEMBL14965806 0.88 MET (0.39) METJAK2JAK1TYK2JAK3
SCHEMBL14965517 0.86 FGFR1 (0.40) MET
SCHEMBL14965570 0.86 JAK2 (0.36) LRRK2METJAK2JAK1TYK2
SCHEMBL14965678 0.84 MTOR (0.37)
SCHEMBL14966317 0.82 LOXL2 (0.42) JAK2JAK3HTR1ADRD2
SCHEMBL14965683 0.82 DRD2 (0.43) HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed