SCHEMBL14967007

SCHEMBL14967007

Fc1cc(Br)ccc1CCOc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.47
NPC1 O15118 3/20 0.45
RAB9A P51151 2/20 0.44
TAAR1 Q96RJ0 1/20 0.43
KCNA3 P22001 1/20 0.42
LTA4H P09960 2/20 0.42
PLA2G2A P14555 1/20 0.42
HPD P32754 2/20 0.42
KDM1A O60341 1/20 0.42
AKR1B1 P15121 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
MAOB P27338 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2236840 0.86 DRD4 (0.49) NPC1RAB9AAKR1B1MEN1KMT2A
SCHEMBL8102862 0.83 NPC1 (0.56) PDPK1NPC1RAB9AHPDKDM1A
SCHEMBL20360954 0.81 MAOB (0.47) NPC1RAB9ATAAR1MEN1KMT2A
SCHEMBL14967099 0.81 KCNA3 (0.42) NPC1RAB9ATAAR1KCNA3LTA4H
SCHEMBL14967564 0.81 ALDH1A1 (0.43) NPC1RAB9ATAAR1KCNA3MEN1
SCHEMBL14966652 0.77 PKM (0.61) RAB9AKMT2A
SCHEMBL20361470 0.76 MAPT (0.43) NPC1RAB9ATAAR1KDM1AMEN1
SCHEMBL12811048 0.76 NPC1 (0.51) PDPK1NPC1TAAR1KDM1AAKR1B1
SCHEMBL27569966 0.76 CHRNB2 (0.44) NPC1RAB9AMEN1KMT2A
SCHEMBL8417765 0.74 KCNA3 (0.61) NPC1RAB9ATAAR1KCNA3LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2780014-A1 MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF Constellation Pharmaceuticals, Inc. (US) 2014-09-24 EP disclosed
WO-2013075083-A1 MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF CONSTELLATION PHARMACEUTICALS (US) 2013-05-23 WO disclosed