SCHEMBL1496969

SCHEMBL1496969

CN1CCN(CCCN(Cc2ccc(C(=O)Nc3cscc3N)nc2)C(=O)NC2=COC=C(C3=CC=CCC3)O2)CC1

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 4/20 0.33
TSHR P16473 2/20 0.32
USP2 O75604 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
MAPT P10636 5/20 0.31
LMNA P02545 2/20 0.31
TP53 P04637 2/20 0.31
THRB P10828 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
KMT2A Q03164 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
ROCK2 O75116 2/20 0.30
HDAC3 O15379 2/20 0.30
HDAC2 Q92769 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1497027 0.96 ALDH1A1 (0.31) TSHRMAPTLMNATP53THRB
SCHEMBL1496990 0.94 USP2 (0.37) TSHRUSP2OPRM1OPRD1MAPT
SCHEMBL2386616 0.93 HDAC1 (0.35) AVPR1ATSHRUSP2SMN1; SMN2MAPT
SCHEMBL1496915 0.92 USP2 (0.36) TSHRUSP2OPRM1OPRD1MAPT
SCHEMBL1497035 0.90 ALDH1A1 (0.37) TSHRUSP2MAPTLMNATP53
SCHEMBL10476409 0.90 TSHR (0.32) AVPR1ATSHRUSP2SMN1; SMN2MAPT
SCHEMBL1497186 0.90 HDAC1 (0.33)
SCHEMBL4217911 0.89 HDAC1 (0.35) TSHRLMNATHRBKDM4EALDH1A1
SCHEMBL1484238 0.88 ROCK1 (0.32) ROCK2HDAC3HDAC2
SCHEMBL4232503 0.86 HSD17B10 (0.40) TSHRUSP2OPRM1OPRD1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2292611-A1 NOVEL THIOPHENEDIAMINE DERIVATIVE HAVING UREA STRUCTURE Santen Pharmaceutical Co., Ltd (JP) 2011-03-09 EP disclosed