SCHEMBL1497035

SCHEMBL1497035

Nc1cscc1NC(=O)c1ccc(CN(CCN2CCOCC2)C(=O)NC2=COC=C(C3=CC=CCC3)O2)cn1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
GAA P10253 3/20 0.37
MAPK1 P28482 2/20 0.37
LMNA P02545 1/20 0.37
THRB P10828 1/20 0.37
POLB P06746 1/20 0.36
TSHR P16473 1/20 0.36
CASR P41180 11/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
ROCK2 O75116 1/20 0.33
ROCK1 Q13464 1/20 0.33
HPGD P15428 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
USP2 O75604 1/20 0.33
TP53 P04637 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
MAPT P10636 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1496990 0.96 USP2 (0.37) ALDH1A1GAALMNATHRBTSHR
SCHEMBL1496915 0.96 USP2 (0.36) ALDH1A1GAAMAPK1LMNATHRB
SCHEMBL1497027 0.94 ALDH1A1 (0.31) ALDH1A1GAAMAPK1LMNATHRB
SCHEMBL1496969 0.90 AVPR1A (0.33) ALDH1A1GAALMNATHRBTSHR
SCHEMBL1496963 0.89 CASR (0.34) ALDH1A1GAAMAPK1LMNATHRB
SCHEMBL4232503 0.89 HSD17B10 (0.40) ALDH1A1GAAMAPK1LMNATHRB
SCHEMBL1497024 0.89 TSHR (0.37) ALDH1A1LMNATHRBTSHRROCK2
SCHEMBL1484238 0.88 ROCK1 (0.32) ROCK2ROCK1
SCHEMBL2386867 0.88 HSD17B10 (0.38) ALDH1A1GAAMAPK1LMNATHRB
SCHEMBL4228734 0.88 HSD17B10 (0.37) ALDH1A1GAAMAPK1LMNATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2292611-A1 NOVEL THIOPHENEDIAMINE DERIVATIVE HAVING UREA STRUCTURE Santen Pharmaceutical Co., Ltd (JP) 2011-03-09 EP disclosed