SCHEMBL14976233

SCHEMBL14976233

CNC(=O)c1c(-c2ccc(F)cc2)nc2sc(-c3csc(C(=O)NC(C)(C)c4ccccc4)c3)cn12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIT P10721 2/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
RAB9A P51151 1/20 0.34
TACR3 P29371 1/20 0.33
MAPT P10636 2/20 0.33
PPARG P37231 1/20 0.33
LMNA P02545 1/20 0.33
EGLN1 Q9GZT9 1/20 0.33
CNR1 P21554 2/20 0.32
CNR2 P34972 2/20 0.32
ROCK2 O75116 1/20 0.32
ROCK1 Q13464 1/20 0.32
ULK1 O75385 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
AURKA O14965 1/20 0.32
DGAT1 O75907 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14977196 0.88 KIT (0.39) KITPTGDR2TACR3SMN1; SMN2DGAT1
SCHEMBL14977224 0.87 KIT (0.39) KITPTGDR2KDM4ENPC1ALDH1A1
SCHEMBL14976444 0.85 CSNK1D (0.39) KITPTGDR2TACR3PPARGROCK2
SCHEMBL14977379 0.82 DGAT2 (0.42) KITPTGDR2KDM4ENPC1MAPT
SCHEMBL14977707 0.82 PPARG (0.39) KITPTGDR2KDM4ENPC1MAPT
SCHEMBL14977623 0.82 PPARG (0.39) KITPTGDR2KDM4ENPC1MAPT
SCHEMBL14977339 0.80 ROCK2 (0.43) KITPTGDR2NPC1MAPTPPARG
SCHEMBL14977718 0.79 ROCK2 (0.35) KITPTGDR2NPC1RAB9ATACR3
SCHEMBL14977301 0.79 CSNK1D (0.36) KITPTGDR2NPC1RAB9ATACR3
SCHEMBL14977582 0.78 CYP2C8 (0.41) CNR1CNR2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013075173-A1 COMPOUNDS FOR THE TREATMENT OF HCV BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2013-05-30 WO disclosed
WO-2013075173-A1 COMPOUNDS FOR THE TREATMENT OF HCV BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2013-05-30 WO disclosed