SCHEMBL14977421

SCHEMBL14977421

CN(C)CCSc1ccc(NS(=O)(=O)c2cccc(C(F)(F)F)c2)cc1F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B2 P37059 1/20 0.52
NR3C1 P04150 1/20 0.47
PGR P06401 1/20 0.47
AR P10275 1/20 0.47
ESR2 Q92731 1/20 0.47
TSHR P16473 1/20 0.46
FFAR1 O14842 1/20 0.46
CDK1 P06493 1/20 0.46
CCNB1 P14635 1/20 0.46
CCNA2 P20248 1/20 0.46
CDK2 P24941 1/20 0.46
CDK7 P50613 1/20 0.46
CCNH P51946 1/20 0.46
CCNA1 P78396 1/20 0.46
FFAR4 Q5NUL3 1/20 0.46
GAA P10253 1/20 0.45
HDAC1 Q13547 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
SERPINE1 P05121 1/20 0.43
PTPN2 P17706 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14976040 0.87 HDAC3 (0.47) PGRFFAR4HDAC1HDAC8PTPN2
SCHEMBL14976775 0.86 HTR6 (0.53) FFAR4GAAKMT2ACACNA1HCACNA1B
SCHEMBL14977115 0.81 HTR6 (0.55) PGRGAAHDAC1HDAC8KMT2A
SCHEMBL14976807 0.81 CA12 (0.49) FFAR1CDK1CCNB1CCNA2CDK2
SCHEMBL14976472 0.80 CACNA1B (0.43) HSD17B2FFAR1FFAR4GAACACNA1H
SCHEMBL13629410 0.77 HSD17B2 (0.61) HSD17B2NR3C1PGRARESR2
SCHEMBL14976733 0.76 HTR7 (0.47) PTPN2PTPN1PTPN5KMT2AHIF1A
SCHEMBL13615168 0.74 HSD17B2 (0.61) HSD17B2NR3C1PGRARESR2
SCHEMBL7572806 0.72 NR3C1 (0.69) HSD17B2NR3C1PGRARESR2
SCHEMBL7573925 0.71 HSD17B2 (0.79) HSD17B2NR3C1PGRARESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013076590-A1 BENZOTHIAZINE COMPOUNDS AS H3 RECEPTOR LIGANDS OXYGEN HEALTHCARE RESEARCH PVT. LTD (IN) 2013-05-30 WO disclosed
WO-2013076590-A1 BENZOTHIAZINE COMPOUNDS AS H3 RECEPTOR LIGANDS OXYGEN HEALTHCARE RESEARCH PVT. LTD (IN) 2013-05-30 WO disclosed