SCHEMBL14999963

SCHEMBL14999963

C=CCCn1c(O[C@@H]2C[C@@H](C(=O)O)N(C(=O)O)C2)cc2ccccc2c1=O

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 5/20 0.33
KAT2B Q92831 1/20 0.32
BTK Q06187 3/20 0.31
LCK P06239 1/20 0.31
SRC P12931 1/20 0.31
KDM4E B2RXH2 2/20 0.31
HSD17B10 Q99714 2/20 0.31
ALDH1A1 P00352 2/20 0.31
POLB P06746 1/20 0.31
HPGD P15428 1/20 0.31
CYP1A2 P05177 2/20 0.31
CNR2 P34972 2/20 0.31
MEN1 O00255 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
KMT2A Q03164 1/20 0.30
ADORA3 P0DMS8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1260139 0.90 KAT2B (0.34) KAT2BBTKLCKSRCKDM4E
SCHEMBL8022909 0.81 P2RX3 (0.41) CNR2
SCHEMBL15000198 0.80 KAT2B (0.32) KAT2BBTKLCKSRCKDM4E
SCHEMBL15000289 0.78
SCHEMBL4246824 0.76 ALDH1A1 (0.44) KDM4EALDH1A1HPGDCYP1A2MEN1
SCHEMBL1260138 0.75 PIM1 (0.39) KAT2BKDM4EHSD17B10ALDH1A1POLB
SCHEMBL15000098 0.72 AGTR2 (0.35) AGTR2
SCHEMBL1260137 0.72 CNR2 (0.32) KDM4EHSD17B10CNR2
SCHEMBL15093160 0.69 SMN1; SMN2 (0.40) KDM4EHSD17B10ALDH1A1CYP1A2MEN1
SCHEMBL17099258 0.69 AGTR2 (0.39) AGTR2KDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2271345-B1 HCV NS3 PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2015-05-20 EP disclosed
US-8461107-B2 HCV NS3 protease inhibitors MERCK SHARP & DOHME CORP. (US) 2013-06-11 US disclosed