SCHEMBL15030636

SCHEMBL15030636

c1ccc(-c2ccc(N3c4cc5c6ccccc6n(-c6ccccc6)c5cc4C4(c5ccccc5Oc5ccccc54)c4cc5c(cc43)c3ccccc3n5-c3ccccc3)cc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ATM Q13315 1/20 0.39
HDAC4 P56524 1/20 0.35
KMT2A Q03164 2/20 0.30
IL1R1 P14778 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15030872 0.97 KDM4E (0.37) L3MBTL1KDM4EATMHDAC4
SCHEMBL16186683 0.92 KDM4E (0.33) L3MBTL1KDM4EATMHDAC4
SCHEMBL15030659 0.89 KDM4E (0.38) L3MBTL1KDM4EATMHDAC4
SCHEMBL15030641 0.89 HDAC4 (0.31) L3MBTL1KDM4EATMHDAC4
SCHEMBL15030690 0.88 KDM4E (0.36) L3MBTL1KDM4EATMHDAC4
SCHEMBL15030792 0.87 KDM4E (0.36) L3MBTL1KDM4EATMHDAC4
SCHEMBL15030846 0.86 KDM4E (0.31) L3MBTL1KDM4EATM
SCHEMBL15030813 0.85 KDM4E (0.32) L3MBTL1KDM4EATM
SCHEMBL19977863 0.84 KDM4E (0.33) L3MBTL1KDM4EATM
SCHEMBL23936688 0.84 L3MBTL1 (0.43) L3MBTL1KDM4EATMHDAC4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10305040-B2 Spiro dihydroacridine derivatives and the use thereof as materials for organic electroluminescence devices MERCK PATENT GMBH (DE) 2019-05-28 US disclosed
EP-2780325-B1 SPIRO-DIHYDROACRIDINE DERIVATIVES AND THEIR USE AS MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2016-02-03 EP disclosed
US-20140316134-A1 SPIRO DIHYDROACRIDINE DERIVATIVES AND THE USE THEREOF AS MATERIALS FOR ORGANIC ELECTROLUMINESCENCE DEVICES MERCK PATENT GMBH (DE) 2014-10-23 US disclosed
US-20140316134-A1 SPIRO DIHYDROACRIDINE DERIVATIVES AND THE USE THEREOF AS MATERIALS FOR ORGANIC ELECTROLUMINESCENCE DEVICES MERCK PATENT GMBH (DE) 2014-10-23 US disclosed
WO-2013083216-A1 SPIRO DIHYDROACRIDINE DERIVATIVES AND THE USE THEREOF AS MATERIALS FOR ORGANIC ELECTROLUMINESCENCE DEVICES MERCK PATENT GMBH (DE) 2013-06-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10305040-B2 Spiro dihydroacridine derivatives and the use thereof as materials for organic electroluminescence devices SORD, ALDH1A1, SDHA L3MBTL1 4454/4885KDM4E 3566/4885ATM 2441/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.