SCHEMBL1503176

SCHEMBL1503176

NC(=O)C1OCc2ccncc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FDPS P14324 1/20 0.36
SIRT3 Q9NTG7 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
ADORA3 P0DMS8 1/20 0.34
TSHR P16473 1/20 0.34
MC4R P32245 1/20 0.34
ADRA1A P35348 1/20 0.34
MC3R P41968 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
CHRNB2 P17787 2/20 0.33
CHRNA4 P43681 2/20 0.33
KDM4C Q9H3R0 2/20 0.33
F7 P08709 1/20 0.33
F3 P13726 1/20 0.33
SARM1 Q6SZW1 1/20 0.33
SIRT2 Q8IXJ6 1/20 0.33
SIRT6 Q8N6T7 1/20 0.33
SIRT1 Q96EB6 1/20 0.33
SIRT5 Q9NXA8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6618609 0.77 ATM (0.42) TSHRALDH1A1KMT2A
SCHEMBL6121157 0.69 DRD2 (0.43) FDPSSIRT3TDP1CYP11B1CYP11B2
SCHEMBL3855349 0.69
SCHEMBL30711624 0.67 SIGMAR1 (0.39) SIRT3TDP1ADORA3TSHRMC4R
SCHEMBL19197111 0.67 NAMPT (0.44) SIRT3TDP1ADORA3TSHRMC4R
SCHEMBL31618283 0.66 CHRNB2 (0.35) FDPSCHRNB2CHRNA4CHRNA7SIGMAR1
SCHEMBL31618365 0.66 CHRNB2 (0.38) FDPSCHRNB2CHRNA4CHRNA7SIGMAR1
SCHEMBL9520473 0.63 ATM (0.35)
SCHEMBL23212526 0.62 MAPT (0.42) FDPSSIRT3TDP1ADORA3TSHR
SCHEMBL31412318 0.62 P2RX7 (0.43) SIRT3TDP1CYP11B1CYP11B2SIRT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2300433-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE Ambrilia Biopharma Inc. (CA) 2011-03-30 EP disclosed
WO-2009146555-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE AMBRILIA BIOPHARMA INC. (CA) 2009-12-10 WO disclosed