SCHEMBL1503319

SCHEMBL1503319

COC(=O)c1ncc(CNCCc2ccc(F)cc2CCOCc2ccccc2)c(CO)c1O

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.38
BCHE P06276 7/20 0.36
KDM4E B2RXH2 3/20 0.35
LMNA P02545 1/20 0.35
NPY1R P25929 1/20 0.35
HTT P42858 1/20 0.35
NPY2R P49146 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MAPT P10636 1/20 0.35
ALDH1A1 P00352 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CD274 Q9NZQ7 2/20 0.34
MEN1 O00255 1/20 0.34
PDCD1 Q15116 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1503317 0.84 KMT2A (0.35) KMT2ABCHEKDM4ELMNANPY1R
SCHEMBL1503138 0.80 KMT2A (0.48) KMT2AKDM4EMAPTALDH1A1L3MBTL1
SCHEMBL1503322 0.76 MAPT (0.34) KMT2ALMNAMAPTALDH1A1L3MBTL1
SCHEMBL1503131 0.75 BCHE (0.39) KMT2ABCHEMEN1
SCHEMBL2221780 0.71 KDM4E (0.47) KMT2AKDM4EALDH1A1L3MBTL1MEN1
SCHEMBL12444364 0.70 ALOX5 (0.40) KMT2AKDM4ELMNAHTTMAPT
SCHEMBL1503187 0.69 ALDH1A1 (0.41) KMT2AKDM4ELMNAMAPTALDH1A1
SCHEMBL1503238 0.67 HDAC1 (0.49) KMT2AKDM4EALDH1A1L3MBTL1
SCHEMBL4306646 0.67 HCAR2 (0.35) KMT2A
SCHEMBL15746784 0.66 BCHE (0.37) KMT2ABCHEMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2300433-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE Ambrilia Biopharma Inc. (CA) 2011-03-30 EP disclosed
WO-2009146555-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE AMBRILIA BIOPHARMA INC. (CA) 2009-12-10 WO disclosed