SCHEMBL1504823

SCHEMBL1504823

COCCOCOc1ccc(C(=O)NC[C@@](C)(C(=O)O)N2CCN(S(=O)(=O)C(C)C)CC2)cc1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
HRH2 P25021 1/20 0.41
HRH1 P35367 1/20 0.41
ADAM17 P78536 5/20 0.40
TP53 P04637 3/20 0.36
MAPT P10636 2/20 0.36
POLB P06746 2/20 0.36
CTNNB1 P35222 1/20 0.36
TSHR P16473 1/20 0.35
CHRM4 P08173 1/20 0.35
PKM P14618 1/20 0.35
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1504784 0.90 ADAM17 (0.43) ALDH1A1HRH2HRH1ADAM17TP53
SCHEMBL1503623 0.85 ALDH1A1 (0.46) ALDH1A1ADAM17TP53POLBCTNNB1
SCHEMBL1504825 0.83 ALDH1A1 (0.45) ALDH1A1HRH2HRH1ADAM17MAPT
SCHEMBL1503650 0.83 ALDH1A1 (0.59) ALDH1A1TP53POLBCTNNB1TSHR
SCHEMBL10275940 0.80 ADAM17 (0.55) HRH2HRH1ADAM17TP53
SCHEMBL10275951 0.80 ADAM17 (0.55) HRH2HRH1ADAM17TP53
SCHEMBL1504822 0.78 ADAM17 (0.51) HRH2HRH1ADAM17TP53
SCHEMBL1504735 0.77 ADAM17 (0.68) ADAM17
SCHEMBL1504939 0.75 ADAM17 (0.60) ALDH1A1ADAM17TP53MAPTPOLB
SCHEMBL1504779 0.74 ADAM17 (0.61) ADAM17CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011033009-A1 N- [2-HYDROXYCARBAMOYL-2- (PIPERAZINYL) ETHYL] BENZAMIDE COMPOUNDS, THEIR PREPARATION AND THEIR USE AS TACE INHIBITORS GALDERMA RESEARCH & DEVELOPMENT (FR) 2011-03-24 WO disclosed