SCHEMBL15047871

SCHEMBL15047871

C#C[C@@H](NC(=O)N1CCOCC1)C1CCCCC1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
CTSS P25774 8/20 0.45
CTSL P07711 3/20 0.44
ALDH1A1 P00352 4/20 0.43
MAPT P10636 3/20 0.43
KMT2A Q03164 1/20 0.43
NPSR1 Q6W5P4 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MCOLN3 Q8TDD5 1/20 0.40
HTT P42858 1/20 0.38
CTSB P07858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15047876 0.77 CTSS (0.56) PKMSMN1; SMN2CTSSCTSLCTSB
SCHEMBL5523635 0.72 PKM (0.48) PKMSMN1; SMN2CTSSCTSLALDH1A1
SCHEMBL8396994 0.72 HTT (0.72) PKMSMN1; SMN2ALDH1A1MAPTKMT2A
SCHEMBL30423567 0.72 HTT (0.72) PKMSMN1; SMN2ALDH1A1MAPTKMT2A
SCHEMBL8392442 0.72 HTT (0.72) PKMSMN1; SMN2ALDH1A1MAPTKMT2A
SCHEMBL27652120 0.70 PKM (0.49) PKMSMN1; SMN2CTSSCTSLALDH1A1
SCHEMBL8395012 0.70 HTT (0.69) PKMSMN1; SMN2ALDH1A1MAPTKMT2A
Bicarbonate SCHEMBL15226014 0.69 HTT (0.68) PKMSMN1; SMN2ALDH1A1MAPTKMT2A
SCHEMBL8392709 0.69 SMN1; SMN2 (0.96) PKMSMN1; SMN2CTSSKMT2AHTT
SCHEMBL12204063 0.69 CTSS (0.59) PKMSMN1; SMN2CTSSCTSLHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8729114-B2 Heteroaryl nitrile compounds useful as inhibitors of Cathepsin-S BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-05-20 US disclosed
US-20130158018-A1 Heteroaryl Nitrile Compounds Useful as Inhibitors of Cathepsin-S BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-06-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130158018-A1 Heteroaryl Nitrile Compounds Useful as Inhibitors of Cathepsin-S CTSS, CTSV, CTSF PKM 4748/4885SMN1; SMN2 2610/4885CTSS 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.